Activation of carboxylic acids by pyrocarbonates: Synthesis of alkylamides of N-protected amino acids

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作者：
Pozdnev, VF
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来源：
BIOORGANICHESKAYA KHIMIYA | 1997年 / 23卷 / 04期
关键词：
amino acids; peptides; alkylamides; di-tert-butyl pyrocarbonate; synthesis; carboxylic group activation;
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摘要：
Alkylamides of amino acids were prepared with high yields via activation of N-protected amino acids by di-tert-pyrocarbonate-pyridine reagent in the presence of alkylamine hydrochlorides and potassium hydrocarbonate.
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页码：262 / 265
页数：4
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