In Vitro and in vivo activity of ARRY-380: A potent, small molecule inhibitor of ErbB2.

被引：0

作者：

Pheneger, Tracy ^{[1
]}

Bouhana, Karyn ^{[1
]}

Anderson, Deborah ^{[1
]}

Garrus, Jennifer ^{[1
]}

Ahrendt, Kateri ^{[1
]}

Allen, Shelley ^{[1
]}

Von Carlowitz, Ira ^{[1
]}

Greschuk, Julie ^{[1
]}

Gross, Stefan ^{[1
]}

Hoffman, Keith ^{[1
]}

Lemieux, Christine ^{[1
]}

Lyssikatos, Joe ^{[1
]}

Callejo, Michele ^{[1
]}

Tarlton, Gene ^{[1
]}

Wallace, Eli ^{[1
]}

Winski, Shannon ^{[1
]}

Woessner, Rich ^{[1
]}

Zhao, Qian ^{[1
]}

Marmsater, Fred ^{[1
]}

Lee, Patrice ^{[1
]}

机构：

[1] Array BioPharma, Boulder, CO USA

来源：

CANCER RESEARCH | 2009年 / 69卷

关键词：

D O I：

暂无

中图分类号：

R73 [肿瘤学];

学科分类号：

100214 ;

摘要：

1795

引用

页数：2

共 50 条

[21] 2-amino-4-methylpyridine as a potent inhibitor of inducible NO synthase activity in vitro and in vivo
Faraci, WS
Nagel, AA
Verdries, KA
Vincent, LA
Xu, H
Nichols, LE
Labasi, JM
Salter, ED
Pettipher, ER
BRITISH JOURNAL OF PHARMACOLOGY, 1996, 119 (06) : 1101 - 1108
[22] A POTENT SMALL MOLECULE PIM KINASE INHIBITOR WITH IN VIVO ORAL AVAILABILITY AND ACTIVITY IN CELL LINES FROM HEMATOLOGICAL MALIGNANCIES
Berk, G.
Gourley, E.
Liu, X. H.
Lamb, J.
Severson, F.
Bearss, J.
Jones, C.
Vankayalapati, H.
Warner, S.
Bearss, D.
HAEMATOLOGICA-THE HEMATOLOGY JOURNAL, 2008, 93 : 113 - 113
[23] Characterization of a Novel, Potent and Selective Small Molecule Spleen Tyrosine Kinase (SYK) Inhibitor in In Vitro and In Vivo Models of Asthma.
Crackower, M. A.
Moy, L. Y.
Jia, Y.
Yu, H.
Vincent, S.
Miller, J. R.
Lieber, G.
Fernandez, X.
Caniga, M.
Gil, M.
Wilhelm, A.
Houshyar, H.
Northrup, A.
Chapman, R.
Abraham, W. M.
Kelly, N.
Hickey, E.
Miller, T.
JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 2012, 129 (02) : AB49 - AB49
[24] IN VITRO AND IN VIVO ANTIVIRAL ACTIVITIES OF AB-423 A POTENT SMALL MOLECULE INHIBITOR OF HEPATITIS B VIRUS CAPSID ASSEMBLY
Mani, N.
Cole, A.
Phelps, J.
Ardzinski, A.
Cobarrubias, K.
Cuconati, A.
Dorsey, B.
Evangelista, E.
Harasym, T.
Kadhim, S.
Lee, A.
Liang, H.
Li, A.
McClintock, K.
Majeski, S.
Reid, S.
Rijnbrand, R.
Tang, S.
Wang, X.
Sofia, M.
JOURNAL OF HEPATOLOGY, 2016, 64 : S392 - S393
[25] In vivo and pharmacodynamic profiling of the KSP inhibitor ARRY-520 supports potent activity in hematological cancers and drug resistant tumors
Woessner, Rich
Cox, April
Koch, Kevin
Lee, Patrice
Rana, Sumeet
Tunquist, Brian
Walker, Duncan
Winkler, Jim
CANCER RESEARCH, 2009, 69
[26] In vitro and in vivo activity of a new small-molecule inhibitor of HDAC6 in mantle cell lymphoma
Perez-Salvia, Montserrat
Aldaba, Eneko
Vara, Yosu
Fabre, Myriam
Ferrer, Cristina
Masdeu, Carme
Zubia, Aizpea
San Sebastian, Eider
Otaegui, Dorleta
Llinas-Arias, Pere
Rossello-Tortella, Margalida
Berdasco, Maria
Moutinho, Catia
Setien, Fernando
Villanueva, Alberto
Gonzalez-Barca, Eva
Muncunill, Josep
Navarro, Jose-Tomas
Piris, Miguel A.
Cossio, Fernando P.
Esteller, Manel
HAEMATOLOGICA, 2018, 103 (11) : E537 - E540
[27] S-222611, a potent, orally active small molecule inhibitor of EGFR and HER2: in vitro kinase inhibition and antitumor activity
Hirata, Michinari
Tanaka, Hidekazu
Dohi, Keiji
Iguchi, Motofumi
Wada, Tohru
Matsuo, Kenji
Kume, Masaharu
Omori, Naoki
Tada, Yukio
Orita, Satoshi
Abe, Kenji
Arimura, Akinori
Matsuo, Yoshiyuki
Kato, Akira
CANCER RESEARCH, 2009, 69
[28] ACC inhibitor demonstrates potent anti-fibrotic activity in vitro and in vivo
Bates, J.
Ghoshal, S.
Wei, L.
Hollenback, D.
Liu, K.
Kusam, S.
Sulfab, M.
Liu, H.
Brockett, R.
Newstrom, D.
Mikaelian, I.
Wang, T.
Harriman, G.
Westlin, W. F.
Rocnik, J.
Harwood, H. J.
Kapeller, R.
Ray, A.
Breckenridge, D.
Fuchs, B. C.
JOURNAL OF HEPATOLOGY, 2018, 68 : S399 - S400
[29] Preclinical characterization of ARRY-575: a potent, selective, and orally bio-available small molecule inhibitor of Chk1
Humphries, M. J.
von Carlowitz, I.
Le Huerou, Y. L.
Randolph, N.
Gunawardana, I.
Mohr, P. J.
Wang, B.
Lyon, M. A.
Chicarelli, M.
Sullivan, F.
Blake, J. F.
Winski, S. L.
Wallace, E.
ANNALS OF ONCOLOGY, 2011, 22 : 23 - 23
[30] A Lipopeptide HIV-1/2 Fusion Inhibitor with Highly Potent In Vitro, Ex Vivo, and In Vivo Antiviral Activity
Chong, Huihui
Xue, Jing
Xiong, Shengwen
Cong, Zhe
Ding, Xiaohui
Zhu, Yuanmei
Liu, Zixuan
Chen, Ting
Feng, Yifan
He, Lei
Guo, Yan
Wei, Qiang
Zhou, Yusen
Qin, Chuan
He, Yuxian
JOURNAL OF VIROLOGY, 2017, 91 (11)

← 1 2 3 4 5 →