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- [31] TAS4464, A Highly Potent and Selective Inhibitor of NEDD8-Activating Enzyme, Suppresses Neddylation and Shows Antitumor Activity in Diverse Cancer ModelsMOLECULAR CANCER THERAPEUTICS, 2019, 18 (07) : 1205 - 1216Yoshimura, Chihoko论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanMuraoka, Hiromi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanOchiiwa, Hiroaki论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanTsuji, Shingo论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanHashimoto, Akihiro论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanKazuno, Hiromi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanNakagawa, Fumio论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanKomiya, Yu论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanSuzuki, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanTakenaka, Toru论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanKumazaki, Masafumi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanFujita, Naoya论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanMizutani, Takashi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, JapanOhkubo, Shuichi论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan Taiho Pharmaceut Co Ltd, Discovery & Preclin Res Div, 3 Okubo, Tsukuba, Ibaraki 3002611, Japan
- [32] The Potent, Highly Selective and Orally Bioavailable Spleen Tyrosine Kinase Inhibitor GSK143 Demonstrates Efficacy in B Cell Receptor and Fc Receptor Signalling in Models of Inflammatory and Autoimmune DiseaseARTHRITIS AND RHEUMATISM, 2012, 64 (10): : S877 - S877Dickson, Marion C.论文数: 0 引用数: 0 h-index: 0机构: GSK, Stevenage, Herts, England GSK, Stevenage, Herts, EnglandSmithers, Nicholas论文数: 0 引用数: 0 h-index: 0机构: GSK, Stevenage, Herts, England GSK, Stevenage, Herts, EnglandLewis, Huw论文数: 0 引用数: 0 h-index: 0机构: GSK, Stevenage, Herts, England GSK, Stevenage, Herts, EnglandRamirez-Molina, Cesar论文数: 0 引用数: 0 h-index: 0机构: GSK, Stevenage, Herts, England GSK, Stevenage, Herts, EnglandMcCleary, Scott论文数: 0 引用数: 0 h-index: 0机构: GSK, Stevenage, Herts, England GSK, Stevenage, Herts, EnglandBarker, Mike论文数: 0 引用数: 0 h-index: 0机构: GSK, Stevenage, Herts, England GSK, Stevenage, Herts, EnglandLiddle, John论文数: 0 引用数: 0 h-index: 0机构: GSK, Stevenage, Herts, England GSK, Stevenage, Herts, England
- [33] E7090, a Novel Selective Inhibitor of Fibroblast Growth Factor Receptors, Displays Potent Antitumor Activity and Prolongs Survival in Preclinical ModelsMOLECULAR CANCER THERAPEUTICS, 2016, 15 (11) : 2630 - 2639Miyano, Saori Watanabe论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Univ Tsukuba, Grad Sch Comprehens Human Sci, Dept Genom Based Drug Discovery, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanYamamoto, Yuji论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanKodama, Kotaro论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanMiyajima, Yukiko论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanMikamoto, Masaki论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanNakagawa, Takayuki论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanKuramochi, Hiroko论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanFunasaka, Setsuo论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanNagao, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanSugi, Naoko Hata论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanOkamoto, Kiyoshi论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanMinoshima, Yukinori论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanNakatani, Yusuke论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanKaroji, Yuki论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanOhashi, Isao论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanYamane, Yoshinobu论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanOkada, Toshimi论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanMatsushima, Tomohiro论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanMatsui, Junji论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanIwata, Masao论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanUenaka, Toshimitsu论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, JapanTsuruoka, Akihiko论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan Eisai & Co Ltd, Tsukuba Res Labs, Tsukuba, Ibaraki, Japan
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- [35] Damage Incorporated: Discovery of the Potent, Highly Selective, Orally Available ATR Inhibitor BAY 1895344 with Favorable Pharmacokinetic Properties and Promising Efficacy in Monotherapy and in Combination Treatments in Preclinical Tumor ModelsJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (13) : 7293 - 7325Luecking, Ulrich论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyWortmann, Lars论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyWengner, Antje M.论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyLefranc, Julien论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyLienau, Philip论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyBriem, Hans论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanySiemeister, Gerhard论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyBoemer, Ulf论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyDenner, Karsten论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanySchaefer, Martina论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyKoppitz, Marcus论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyEis, Knut论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyBartels, Florian论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyBader, Benjamin论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyBone, Wilhelm论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyMoosmayer, Dieter论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyHolton, Simon J.论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyEberspaecher, Uwe论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyGrudzinska-Goebel, Joanna论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanySchatz, Christoph论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyDeeg, Gesa论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, GermanyMumberg, Dominik论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germanyvon Nussbaum, Franz论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany Bayer AG, Res & Dev, Pharmaceut, D-13353 Berlin, Germany
- [36] K0706, A Potent Orally Bioavailable Brain-Penetrating Selective Inhibitor of cABL Protein Tyrosine Kinase, Exhibits Neuroprotective Activity in Preclinical Models of Parkinson's DiseaseMOVEMENT DISORDERS, 2019, 34Mandhane, S.论文数: 0 引用数: 0 h-index: 0Soni, D.论文数: 0 引用数: 0 h-index: 0Jani, K.论文数: 0 引用数: 0 h-index: 0Sengupta, P.论文数: 0 引用数: 0 h-index: 0Patel, A.论文数: 0 引用数: 0 h-index: 0Bambal, R.论文数: 0 引用数: 0 h-index: 0Ramanathan, V.论文数: 0 引用数: 0 h-index: 0Zala, Y.论文数: 0 引用数: 0 h-index: 0Dharmadhikari, N.论文数: 0 引用数: 0 h-index: 0Rao, C.论文数: 0 引用数: 0 h-index: 0Raghavan, A.论文数: 0 引用数: 0 h-index: 0Damle, N.论文数: 0 引用数: 0 h-index: 0
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