Understanding 5-aminosalicylic acid (5-ASA) release profiles from pH-Dependent delayed-release formulations: a Multidisciplinary approach

被引:0
|
作者
Tenjarla, Srini [1 ]
Karlstadt, Robyn [1 ]
Joseph, Raymond [1 ]
机构
[1] Shire Pharmaceut Inc, Wayne, PA USA
来源
关键词
D O I
10.14309/00000434-200809001-01113
中图分类号
R57 [消化系及腹部疾病];
学科分类号
摘要
1113
引用
收藏
页码:S435 / S435
页数:1
相关论文
共 50 条
  • [31] PHARMACOKINETICS OF 5-AMINOSALICYLIC ACID FROM CONTROLLED-RELEASE CAPSULES IN MAN
    YU, DK
    MORRILL, B
    EICHMEIER, LS
    LANMAN, RC
    LANMAN, MB
    GIESING, DH
    WEIR, SJ
    EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1995, 48 (3-4) : 273 - 277
  • [32] Systemic availability of 5-aminosalicylic acid: Comparison of delayed release and an azo-bond preparation
    Gionchetti, P
    Campieri, M
    Venturi, A
    Rizzello, F
    Ferretti, M
    Brignola, C
    Miglioli, M
    ALIMENTARY PHARMACOLOGY & THERAPEUTICS, 1996, 10 (04) : 601 - 605
  • [33] A DELAYED RELEASE 5-AMINOSALICYLIC ACID TABLET FORMULATION FOR THE TREATMENT OF INFLAMMATORY BOWEL-DISEASE
    HEALEY, JNC
    HARDY, JG
    REYNOLDS, JR
    GASTROENTEROLOGY, 1987, 92 (05) : 1429 - 1429
  • [34] Predicting Regional Colonic Concentrations of 5-Aminosalicylic Acid (5-ASA) From Oral and Topical Therapy With Dynamic Modeling in Ulcerative Colitis
    Stobaugh, Derrick J.
    Deepak, Parakkal
    Hannon, Bruce
    Ehrenpreis, Eli D.
    GASTROENTEROLOGY, 2012, 142 (05) : S389 - S389
  • [35] INFLUENCE OF HYDROPHILIC ADDITIVES ON 5-AMINOSALICYLIC ACID RELEASE RATE FROM MATRIX PELLETS
    DEBRANT, V
    REMON, JP
    5TH INTERNATIONAL CONFERENCE ON PHARMACEUTICAL TECHNOLOGY, VOLS 1-5, 1989, : 222 - 230
  • [36] Release of 5-ASA from Asacol appears independent of gut luminal pH in ulcerative colitis
    Nugent, S
    Rampton, D
    Obeid, O
    Evans, D
    Kumar, D
    GASTROENTEROLOGY, 2001, 120 (05) : A455 - A455
  • [37] 5-Aminosalicylic Acid and its major metabolite levels in patients with moderately active ulcerative Colitis following oral administration of delayed-release Mesalamine tablets
    Sandborn, W.
    Balan, G.
    Ajayi, F.
    INFLAMMATORY BOWEL DISEASES, 2008, 14 (12) : S30 - S30
  • [38] Controlled release of 5-aminosalicylic acid from a new pH responsive polymer derived from tamarind seed polysaccharide, acrylic acid, and polyamidoamine
    Dey, R. K.
    Tiwary, G. S.
    Patnaik, Tanushree
    Jha, Usha
    POLYMER BULLETIN, 2011, 66 (05) : 583 - 598
  • [39] Controlled release of 5-aminosalicylic acid from a new pH responsive polymer derived from tamarind seed polysaccharide, acrylic acid, and polyamidoamine
    R. K. Dey
    G. S. Tiwary
    Tanushree Patnaik
    Usha Jha
    Polymer Bulletin, 2011, 66 : 583 - 598
  • [40] Concentration Dependence of 5-Aminosalicylic Acid Pharmacological Actions in Intestinal Mucosa after Oral Administration of a pH-Dependent Formulation
    Hirayama, Masamichi
    Toda, Ryoko
    Ozaki, Tomoko
    Hasegawa, Junko
    Nakamura, Toshifumi
    Naraki, Yoko
    Haraguchi, Yukari
    Hori, Yuko
    Tanaka, Takao
    Takei, Mineo
    Mera, Yukinori
    Yoshii, Kazuyoshi
    Kawabata, Yoshihiro
    MOLECULAR PHARMACEUTICS, 2011, 8 (04) : 1083 - 1089