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- [41] Fragment-based approach to covalent inhibitors of catalytic cysteinesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 246Kathman, Stefan论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Evanston, IL 60208 USA Northwestern Univ, Dept Chem, Evanston, IL 60208 USAXu, Ziyang论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Evanston, IL 60208 USA Northwestern Univ, Dept Chem, Evanston, IL 60208 USAStatsyuk, Alexander论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Dept Chem, Evanston, IL 60208 USA Northwestern Univ, Dept Chem, Evanston, IL 60208 USA
- [42] Fragment-based discovery of focal adhesion kinase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (19) : 5401 - 5409Graedler, Ulrich论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyBomke, Joerg论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyMusil, Djordje论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyDresing, Verena论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyLehmann, Martin论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyHoelzemann, Guenter论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyGreiner, Hartmut论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyEsdar, Christina论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyKrier, Mireille论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, GermanyHeinrich, Timo论文数: 0 引用数: 0 h-index: 0机构: Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany Merck Serono Res, Merck KGaA, D-64293 Darmstadt, Germany
- [43] Fragment-based approach to developing histidine kinase inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251Wassarman, Douglas论文数: 0 引用数: 0 h-index: 0机构: Williams Coll, Williamstown, MA 01267 USA Williams Coll, Williamstown, MA 01267 USAHuang, Tony论文数: 0 引用数: 0 h-index: 0机构: Williams Coll, Williamstown, MA 01267 USA Williams Coll, Williamstown, MA 01267 USABlair, Jimmy论文数: 0 引用数: 0 h-index: 0机构: Williams Coll, Dept Chem, Williamstown, MA 01267 USA Williams Coll, Williamstown, MA 01267 USA
- [44] Fragment-Based Design of Mycobacterium tuberculosis InhA InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (09) : 4749 - 4761Sabbah, Mohamad论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandMendes, Vitor论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandVistal, Robert G.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandDias, David M. G.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandZahorszka, Monika论文数: 0 引用数: 0 h-index: 0机构: Comenius Univ, Dept Biochem, Fac Nat Sci, Bratislava 84215, Slovakia Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandMikusova, Katarina论文数: 0 引用数: 0 h-index: 0机构: Comenius Univ, Dept Biochem, Fac Nat Sci, Bratislava 84215, Slovakia Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandKordulakova, Jana论文数: 0 引用数: 0 h-index: 0机构: Comenius Univ, Dept Biochem, Fac Nat Sci, Bratislava 84215, Slovakia Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandCoyne, Anthony G.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandBlundell, Tom L.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Biochem, Cambridge CB2 1GA, England Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandAbell, Chris论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England Univ Cambridge, Dept Chem, Cambridge CB2 1EW, England
- [45] Fragment-based Identification of Hsp90 InhibitorsCHEMMEDCHEM, 2009, 4 (06) : 963 - 966Barker, John J.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandBarker, Oliver论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandBoggio, Roberto论文数: 0 引用数: 0 h-index: 0机构: Congenia Srl, Genextra Grp, I-20139 Milan, Italy Evotec, Abingdon OX10 4SA, Oxon, EnglandChauhan, Viddhata论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandCheng, Robert K. Y.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandCorden, Vincent论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandCourtney, Stephen M.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandEdwards, Neil论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandFalque, Virginie M.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandFusar, Fulvia论文数: 0 引用数: 0 h-index: 0机构: DAC Srl, Genextra Grp, I-20139 Milan, Italy Evotec, Abingdon OX10 4SA, Oxon, EnglandGardiner, Mihaly论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandHamelin, Estelle M. N.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandHesterkamp, Thomas论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandIchihara, Osamu论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandJones, Richard S.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandMather, Owen论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandMercurio, Ciro论文数: 0 引用数: 0 h-index: 0机构: DAC Srl, Genextra Grp, I-20139 Milan, Italy Evotec, Abingdon OX10 4SA, Oxon, England论文数: 引用数: h-index:机构:Montalbetti, Christian A. G. N.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandMueller, Annett论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandPatel, Deepti论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandPhillips, Banu G.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandVarasi, Mario论文数: 0 引用数: 0 h-index: 0机构: DAC Srl, Genextra Grp, I-20139 Milan, Italy Evotec, Abingdon OX10 4SA, Oxon, EnglandWhittaker, Mark论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandWinkler, Dirk论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, EnglandYarnold, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Evotec, Abingdon OX10 4SA, Oxon, England Evotec, Abingdon OX10 4SA, Oxon, England
- [46] Discovery of KATII inhibitors via a fragment-based approachABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251Han, Ying论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAStachura, Sylwia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAMcClure, Andrea论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USACavallaro, Cullen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAAllard, Christopher论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USARajamani, Ramkumar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAYong, Wei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USALewis, Hal论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAMuckelbauer, Jodi论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USALoughney, Deborah论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAMetzler, William论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USANirschl, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAWeller, Harold论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, LVL, Princeton, NJ USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USAGerritz, Sam论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, 5 Res Pkwy, Wallingford, CT 06492 USA
- [47] Fragment-Based Discovery of Inhibitors of Protein Kinase BCURRENT TOPICS IN MEDICINAL CHEMISTRY, 2009, 9 (18) : 1705 - 1717Davies, Thomas G.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Inst Canc Res, Canc Res UK Ctr Canc Therapeut, Sutton SM2 5NG, Surrey, EnglandWoodhead, Steven J.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Inst Canc Res, Canc Res UK Ctr Canc Therapeut, Sutton SM2 5NG, Surrey, EnglandCollins, Ian论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Ctr Canc Therapeut, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Ctr Canc Therapeut, Sutton SM2 5NG, Surrey, England
- [48] Identification of potent, selective JAK2 inhibitors using a fragment-based screening approachEJC SUPPLEMENTS, 2008, 6 (12): : 180 - 180Wallis, N. G.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Biol, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandChessari, G.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Computat Chem, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandCurry, J. E.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Biol, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandHamlett, C.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Chem, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandLewry, K. A.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Biol, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandLyons, J.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Biol, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandRichardson, C. J.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Biol, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandTisi, D.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Struct Biol, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandWalker, D.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Chem, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, EnglandWoodhead, A. J.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Chem, Cambridge, England Astex Therapeut Ltd, Biol, Cambridge, England
- [49] Efficient exploration of chemical space by fragment-based screeningPROGRESS IN BIOPHYSICS & MOLECULAR BIOLOGY, 2014, 116 (2-3): : 82 - 91Hall, Richard J.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandMortenson, Paul N.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandMurray, Christopher W.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, England
- [50] Fragment-based development of bacterial DsbA inhibitors as novel anti-virulence agentsACTA CRYSTALLOGRAPHICA A-FOUNDATION AND ADVANCES, 2021, 77 : C567 - C567Wang, Geqing论文数: 0 引用数: 0 h-index: 0机构: La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaAlwan, Wesam论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaBentley, Matthew论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaMohanty, Biswaranjan论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaDoak, Bradley论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaDhouib, Rabeb论文数: 0 引用数: 0 h-index: 0机构: Queensland Univ Technol, Inst Hlth & Biomed Innovat, Kelvin Grove, Qld 4059, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, Australia论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Capuano, Benvenuto论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaScammells, Peter论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaMartin, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Griffith Univ, Griffith Inst Drug Discovery, Nathan, Qld 4111, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, AustraliaScanlon, Martin论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Monash Inst Pharmaceut Sci, Med Chem, Parkville, Vic 3052, Australia La Trobe Univ, La Trobe Inst Mol Sci, Dept Biochem & Genet, Bundoora, Vic 3086, Australia论文数: 引用数: h-index:机构: