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- [21] Discovery of a Potent and Selective ROMK Inhibitor with Pharmacokinetic Properties Suitable for Preclinical EvaluationACS MEDICINAL CHEMISTRY LETTERS, 2015, 6 (07): : 747 - 752Walsh, Shawn P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAShahripour, Aurash论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USATang, Haifeng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USATeumelsan, Nardos论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAFrie, Jessica论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAZhu, Yuping论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAPriest, Birgit T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USASwensen, Andrew M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USALiu, Jessica论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAMargulis, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAVisconti, Richard论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAWeinglass, Adam论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAFelix, John P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USABrochu, Richard M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USABailey, Timothy论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAThomas-Fowlkes, Brande论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAAlonso-Galicia, Magdalena论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAZhou, Xiaoyan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAPai, Lee-Yuh论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USACorona, Aaron论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAHampton, Caryn论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAHernandez, Melba论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USABentley, Ross论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAChen, Jing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAShah, Kashmira论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAMetzger, Joseph论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAForrest, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAOwens, Karen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Pharmacokinet Pharmacodynam & Drug Metab, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USATong, Vincent论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Pharmacokinet Pharmacodynam & Drug Metab, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAHa, Sookhee论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Modeling & Informat, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USARoy, Sophie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAKaczorowski, Gregory J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAYang, Lihu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAParmee, Emma论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAGarcia, Maria L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USASullivan, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Cardiometab Dis, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USAPasternak, Alexander论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Discovery Chem, Kenilworth, NJ 07033 USA
- [22] Discovery of a potent and selective Axl inhibitor in preclinical modelBIOORGANIC & MEDICINAL CHEMISTRY, 2021, 39Inoue, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanYamane, Yoshinobu论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanTsukamoto, Shuntaro论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanAzuma, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanNagao, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanMurai, Norio论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanNishibata, Kyoko论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanFukushima, Sayo论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanIchikawa, Kenji论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanNakagawa, Takayuki论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanSugi, Naoko Hata论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanIto, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanKato, Yu论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanGoto, Aya论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Drug Safety, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanKakiuchi, Dai论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Drug Safety, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanUeno, Takashi论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Drug Metab & Pharmacokinet, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanMatsui, Junji论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Biopharmacol, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, JapanMatsushima, Tomohiro论文数: 0 引用数: 0 h-index: 0机构: Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan Eisai & Co Ltd, Med Chem, Tsukuba Res Labs, 5-1-3 Tokodai, Tsukuba, Ibaraki 3002635, Japan
- [23] Discovery of a novel and highly selective CDK9 kinase inhibitor (JSH-009) with potent antitumor efficacy in preclinical acute myeloid leukemia modelsInvestigational New Drugs, 2020, 38 : 1272 - 1281Li Wang论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyChen Hu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyAoli Wang论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyCheng Chen论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyJiaxin Wu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyZongru Jiang论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyFengming Zou论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyKailin Yu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyHong Wu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyJuan Liu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyWenliang Wang论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyZuowei Wang论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyBeilei Wang论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyZiping Qi论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyQingwang Liu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyWenchao Wang论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyLili Li论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyJian Ge论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyJing Liu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical BiologyQingsong Liu论文数: 0 引用数: 0 h-index: 0机构: Hefei Institutes of Physical Science,High Magnetic Field Laboratory, Key Laboratory of High Magnetic Field and Ion Beam Physical Biology
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