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- [1] Discovery and preclinical evaluation of a novel highly selective and potent CDK12 inhibitorCANCER SCIENCE, 2023, 114 : 831 - 831Yamakawa, Hiroko论文数: 0 引用数: 0 h-index: 0机构: Chordia Therapeut Inc, Fujisawa, Kanagawa, Japan Chordia Therapeut Inc, Fujisawa, Kanagawa, JapanMizutani, Akio论文数: 0 引用数: 0 h-index: 0机构: Chordia Therapeut Inc, Fujisawa, Kanagawa, Japan Chordia Therapeut Inc, Fujisawa, Kanagawa, JapanArikawa, Yasuyoshi论文数: 0 引用数: 0 h-index: 0机构: Chordia Therapeut Inc, Fujisawa, Kanagawa, Japan Chordia Therapeut Inc, Fujisawa, Kanagawa, JapanEbara, Shunsuke论文数: 0 引用数: 0 h-index: 0机构: Chordia Therapeut Inc, Fujisawa, Kanagawa, Japan Chordia Therapeut Inc, Fujisawa, Kanagawa, JapanSatoh, Yoshihiko论文数: 0 引用数: 0 h-index: 0机构: Chordia Therapeut Inc, Fujisawa, Kanagawa, Japan Chordia Therapeut Inc, Fujisawa, Kanagawa, JapanMorishita, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Chordia Therapeut Inc, Fujisawa, Kanagawa, Japan Chordia Therapeut Inc, Fujisawa, Kanagawa, Japan
- [2] Discovery of a highly potent and selective dual PROTAC degrader of CDK12 and CDK13CANCER RESEARCH, 2023, 83 (07)Chang, Yu论文数: 0 引用数: 0 h-index: 0Yang, Jianzhang论文数: 0 引用数: 0 h-index: 0Tien, Jean Ching-Yi论文数: 0 引用数: 0 h-index: 0Wang, Zhen论文数: 0 引用数: 0 h-index: 0Zhou, Yang论文数: 0 引用数: 0 h-index: 0Zhang, Pujuan论文数: 0 引用数: 0 h-index: 0Huang, Weixue论文数: 0 引用数: 0 h-index: 0Vo, Josh论文数: 0 引用数: 0 h-index: 0Apel, Ingrid J.论文数: 0 引用数: 0 h-index: 0Wang, Cynthia论文数: 0 引用数: 0 h-index: 0Zeng, Victoria Zhixuan论文数: 0 引用数: 0 h-index: 0Cheng, Yunhui论文数: 0 引用数: 0 h-index: 0Li, Shuqin论文数: 0 引用数: 0 h-index: 0Wang, George Xiaoju论文数: 0 引用数: 0 h-index: 0Ding, Ke论文数: 0 引用数: 0 h-index: 0Chinnaiyan, Arul M.论文数: 0 引用数: 0 h-index: 0
- [3] Discovery of a Highly Potent and Selective Dual PROTAC Degrader of CDK12 and CDK13JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (16) : 11066 - 11083Yang, Jianzhang论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaChang, Yu论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaTien, Jean Ching-Yi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaWang, Zhen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Bioorgan & Nat Prod Chem, Shanghai 200032, Peoples R China Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaZhou, Yang论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaZhang, Pujuan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Bioorgan & Nat Prod Chem, Shanghai 200032, Peoples R China Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaHuang, Weixue论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Bioorgan & Nat Prod Chem, Shanghai 200032, Peoples R China Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaVo, Josh论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaApel, Ingrid J.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaWang, Cynthia论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaZeng, Victoria Zhixuan论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaCheng, Yunhui论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaWang, George Xiaoju论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Computat Med & Bioinformat, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaChinnaiyan, Arul M.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Howard Hughes Med Inst, Dept Pathol, Dept Computat Med & Bioinformat, Ann Arbor, MI 48109 USA Univ Michigan, Dept Urol, Ann Arbor, MI 48109 USA Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R ChinaDing, Ke论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Bioorgan & Nat Prod Chem, Shanghai 200032, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Bioorgan & Nat Prod Chem, Shanghai 200032, Peoples R China Chinese Acad Sci, Inst Basic Med & Canc IBMC, Hangzhou 310022, Zhejiang, Peoples R China Jinan Univ, Affiliated Hosp 1, Huaqiao Hosp, Guangzhou 510632, Peoples R China Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China
- [4] Preclinical evaluation of PD and efficacy of novel potent selective and orally bioavailable CDK12 covalent inhibitors in TNBC modelCANCER RESEARCH, 2018, 78 (13)Poddutoori, Ramulu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaRajagopalan, Sujatha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaMukherjee, Subhendu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaMarappan, Sivapriya论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSamiulla, D. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSivakumar, Sasirekha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaNayak, Shilpa S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaRavindra, M., V论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaMurtuza, Hadianawala论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDevaraja, T. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaKondela, Srinivas论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaTgore, Suraj论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDhudashiya, Amit A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaCharamanna, K. B.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaAntony, Thomas论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaDaginakatte, Girish论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaGiri, Sanjeev论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaChelur, Shekar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaRamachandra, Murali论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaPandit, Chetan论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, IndiaSamajdar, Susanta论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India
- [5] Discovery of YJZ5118: A Potent and Highly Selective Irreversible CDK12/13 Inhibitor with Synergistic Effects in Combination with Akt InhibitionJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (06) : 6718 - 6734Yang, Jianzhang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaChang, Yu论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaZhou, Kaijie论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaHuang, Weixue论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaTien, Jean Ching-Yi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaZhang, Pujuan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaLiu, Wenyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaZhou, Licheng论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaZhou, Yang论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Coll Pharm, Int Cooperat Lab Tradit Chinese Med Modernizat, Guangzhou City Key Lab Precis Chem Drug Dev, Guangzhou 511400, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaRen, Xiaomei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaMannan, Rahul论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaMahapatra, Somnath论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaZhang, Yuping论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaHamadeh, Rudana论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaErvine, Grafton论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaWang, Zhen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaWang, George Xiaoju论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaChinnaiyan, Arul M.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Michigan Ctr Translat Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Howard Hughes Med Inst, Ann Arbor, MI 48109 USA Univ Michigan, Dept Urol, Ann Arbor, MI 48109 USA Univ Michigan, Rogel Canc Ctr, Ann Arbor, MI 48109 USA Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R ChinaDing, Ke论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, Shanghai 200032, Peoples R China
- [6] Preclinical characterization of LY3537982, a novel, highly selective and potent KRAS-G12C inhibitor.CANCER RESEARCH, 2021, 81 (13)Peng, Sheng-Bin论文数: 0 引用数: 0 h-index: 0机构: Lilly, Loxo Oncol, Indianapolis, IN USA Lilly, Loxo Oncol, Indianapolis, IN USASi, Chong论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAZhang, Youyan论文数: 0 引用数: 0 h-index: 0机构: Lilly, Loxo Oncol, Indianapolis, IN USA Lilly, Loxo Oncol, Indianapolis, IN USAVan Horn, Robert D.论文数: 0 引用数: 0 h-index: 0机构: Lilly, Loxo Oncol, Indianapolis, IN USA Lilly, Loxo Oncol, Indianapolis, IN USALin, Xi论文数: 0 引用数: 0 h-index: 0机构: Lilly, Loxo Oncol, Indianapolis, IN USA Lilly, Loxo Oncol, Indianapolis, IN USAGong, Xueqian论文数: 0 引用数: 0 h-index: 0机构: Lilly, Loxo Oncol, Indianapolis, IN USA Lilly, Loxo Oncol, Indianapolis, IN USAHuber, Lysiane论文数: 0 引用数: 0 h-index: 0机构: Lilly, Loxo Oncol, Indianapolis, IN USA Lilly, Loxo Oncol, Indianapolis, IN USADonoho, Gregory论文数: 0 引用数: 0 h-index: 0机构: Lilly, Loxo Oncol, Indianapolis, IN USA Lilly, Loxo Oncol, Indianapolis, IN USACurtis, Carmen论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAStrelow, John M.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USABocchinfuso, Wayne P.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAGuo, Deqi论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USABoulet, Serge L.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USABarda, David论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAManglicmot, Danalyn论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, San Diego, CA USA Lilly, Loxo Oncol, Indianapolis, IN USASaflor, Melbert-Brian D.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, San Diego, CA USA Lilly, Loxo Oncol, Indianapolis, IN USAWang, Jing论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, San Diego, CA USA Lilly, Loxo Oncol, Indianapolis, IN USAXiao, Junpeng论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAChalmers, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USABurns, Lee论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USALinder, Ryan J.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAAckermann, Bradley L.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USACornwell, Paul D.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAZhou, Lian论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAMcCann, Denis论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USAHenry, James论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Lilly, Loxo Oncol, Indianapolis, IN USA
- [7] Discovery and evaluation of ISM6466A, a novel covalent CDK12 inhibitor for the treatment of cancerCANCER RESEARCH, 2023, 83 (07)Min, Lihua论文数: 0 引用数: 0 h-index: 0Lu, Hongfu论文数: 0 引用数: 0 h-index: 0Zhang, Yihong论文数: 0 引用数: 0 h-index: 0Wu, Jianping论文数: 0 引用数: 0 h-index: 0Cai, Xin论文数: 0 引用数: 0 h-index: 0Zheng, Min论文数: 0 引用数: 0 h-index: 0Cui, Hui论文数: 0 引用数: 0 h-index: 0Qiao, Junwen论文数: 0 引用数: 0 h-index: 0Ding, Xiao论文数: 0 引用数: 0 h-index: 0Rao, Sujata论文数: 0 引用数: 0 h-index: 0Ren, Feng论文数: 0 引用数: 0 h-index: 0Zhavoronkov, Alex论文数: 0 引用数: 0 h-index: 0
- [8] Discovery and Biological Evaluation of a Novel Highly Potent Selective Butyrylcholinsterase InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (17) : 10030 - 10044Li, Qi论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaXing, Shuaishuai论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaChen, Ying论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLiao, Qinghong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaXiong, Baichen论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaHe, Siyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Jiangsu Key Lab Carcinogenesis & Intervent, Sch Basic Med & Clin Pharm, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLu, Weixuan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLiu, Yang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaYang, Hongyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLi, Qihang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaFeng, Feng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Nat Med Chem, Nanjing 211198, Peoples R China Jiangsu Food & Pharmaceut Sci Coll, Huaian 223003, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaLiu, Wenyuan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaChen, Yao论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R ChinaSun, Haopeng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Pharm, Nanjing 211198, Peoples R China
- [9] Potent selective and orally bioavailable inhibition of CDK12 by novel covalent inhibitorsMOLECULAR CANCER THERAPEUTICS, 2018, 17 (01)Poddutoori, Ramulu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaRajagopalan, Sujatha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaMukherjee, Subhendu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaMarappan, Sivapriya论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaSamiulla, D. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaKasturi, Venkateswarlu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaSivakumar, Sasirekha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaNayak, Shilpa论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaRavindra, M., V论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaTgore, Suraj论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaDhudashiya, Amit论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaCharamanna, K. B.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaAntony, Thomas论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaMahaboobi, M.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaGiri, Sanjeev论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaDaginakatte, Girish C.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaChelur, Shekar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaRamachandra, Murali论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaPandit, Chetan论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, IndiaSamajdar, Susanta论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol, Bangalore, Karnataka, India Aurigene Discovery Technol, Bangalore, Karnataka, India
- [10] Discovery and resistance mechanism of a selective CDK12 degraderNATURE CHEMICAL BIOLOGY, 2021, 17 (06) : 675 - 683Jiang, Baishan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGao, Yang论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAChe, Jianwei论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USALu, Wenchao论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAKaltheuner, Ines H.论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Inst Struct Biol, Bonn, Germany Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USADries, Ruben论文数: 0 引用数: 0 h-index: 0机构: Boston Univ, Dept Hematol & Oncol, Boston, MA 02215 USA Boston Univ, Dept Computat Med, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAKalocsay, Marian论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Lab Syst Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USABerberich, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Lab Syst Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAJiang, Jie论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAYou, Inchul论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAKwiatkowski, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USARiching, Kristin M.论文数: 0 引用数: 0 h-index: 0机构: Promega Corp, Madison, WI USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USADaniels, Danette L.论文数: 0 引用数: 0 h-index: 0机构: Promega Corp, Madison, WI USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USASorger, Peter K.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Lab Syst Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGeyer, Matthias论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Inst Struct Biol, Bonn, Germany Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAZhang, Tinghu论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA