Novel Pyrazolopyridine Inhibitors of Monoacylglycerol Lipase for the Treatment of Neurodegenerative Diseases and Neuroinflammation

被引:1
|
作者
Rosse, Gerard [1 ]
机构
[1] Arrival Discovery LLC, San Diego, CA 92128 USA
来源
ACS MEDICINAL CHEMISTRY LETTERS | 2024年 / 15卷 / 01期
关键词
D O I
10.1021/acsmedchemlett.3c00548
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
This work highlights the use of bicyclic heterocyclic compounds as monoacylglycerol lipase inhibitors potentially in the treatment of Alzheimer's disease, Parkinson's disease, ALS, traumatic brain injury, and multiple sclerosis.
引用
收藏
页码:19 / 20
页数:2
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