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- [11] HJM-353: A potent, selective and orally bioavailable EED inhibitor with robust anti-tumor activitiesANNALS OF ONCOLOGY, 2022, 33 (07) : S1122 - S1122Ma, X.论文数: 0 引用数: 0 h-index: 0机构: Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R China Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R ChinaQi, W.论文数: 0 引用数: 0 h-index: 0机构: ShanghaiTech Univ, Res Dept, Zhangjiang Campus, Shanghai, Peoples R China Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R ChinaDu, Y.论文数: 0 引用数: 0 h-index: 0机构: Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R China Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R ChinaKong, D.论文数: 0 引用数: 0 h-index: 0机构: Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R China Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R ChinaGeng, Y.论文数: 0 引用数: 0 h-index: 0机构: Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R China Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R ChinaZeng, L.论文数: 0 引用数: 0 h-index: 0机构: Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R China Jing Med Technol Shanghai Ltd, Res Dept, Shanghai, Peoples R China
- [12] Structure-Activity Relationship of Potent, Selective, and Orally Bioavailable Molecular Glue Degraders of CK1αACS MEDICINAL CHEMISTRY LETTERS, 2024, 15 (10): : 1692 - 1698Nishiguchi, Gisele论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USACaine, Elizabeth A.论文数: 0 引用数: 0 h-index: 0机构: Promega Corp, Madison, WI 53711 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAMcgowan, Kevin论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAShi, Zhe论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAAggarwal, Anup论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAMayasundari, Anand论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAPrice, Jeanine论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAYang, Lei论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USALi, Yong论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAFu, Xiang论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAMascibroda, Lauren G.论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Pathol, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USADas, Sourav论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USADaniels, Danette L.论文数: 0 引用数: 0 h-index: 0机构: Foghorn Therapeut Inc, Cambridge, MA 02139 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAUrh, Marjeta论文数: 0 引用数: 0 h-index: 0机构: Promega Corp, Madison, WI 53711 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USAKlco, Jeffery M.论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Pathol, Memphis, TN 38105 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USARiching, Kristin M.论文数: 0 引用数: 0 h-index: 0机构: Promega Corp, Madison, WI 53711 USA St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USARankovic, Zoran论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA Inst Canc Res, Ctr Prot Degradat, Sutton SM2 5NG, England St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA
- [13] Discovery of novel, potent, and orally bioavailable HDACs inhibitors with LSD1 inhibitory activity for the treatment of solid tumorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 254Duan, Yingchao论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaYu, Tong论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaJin, Linfeng论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZhang, Shaojie论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaShi, Xiaojing论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Acad Med Sci, Lab Anim Ctr, Zhengzhou 450052, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZhang, Yizhe论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZhou, Nanqian论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ Peoples Hosp, Henan Univ Peoples Hosp, Henan Prov Peoples Hosp, Dept Ultrasonog, Zhengzhou 450003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaXu, Yongtao论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Med Engn, Henan Int Joint Lab Neural Informat Anal & Drug In, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaLu, Wenfeng论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Med Engn, Henan Int Joint Lab Neural Informat Anal & Drug In, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZhou, Huimin论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaZhu, Huijuan论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaBai, Suping论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaHu, Kua论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R ChinaGuan, Yuanyuan论文数: 0 引用数: 0 h-index: 0机构: Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China Xinxiang Med Univ, Sch Pharm, Xinxiang 453003, Henan, Peoples R China
- [14] Synergistic Combination Activity of the Novel GSPT1 Degrader CC-90009 in Acute Myeloid Leukemia ModelsBLOOD, 2021, 138Pierce, Daniel W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAYao, Tsun-Wen Sheena论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Formerly ONC TRC, San Diego, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAYao, Sheena论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Formerly ONC TRC, San Diego, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAPace, Emily论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Formerly ONC TRC, San Diego, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAWang, Hongbin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAFlandin-Blety, Pierre论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USABenitez, Alicia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, BMS Ctr Innovat & Translat Res Europe CITRE, ONC TRC, Seville, Spain Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAGuarinos, Carla论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, BMS Ctr Innovat & Translat Res Europe CITRE, ONC TRC, Seville, Spain Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAHoffmann, Matthew论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Princeton, NJ USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USACarrancio, Soraya论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAFan, Jonhong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Formerly ONC TRC, San Diego, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USAPourdehnad, Michael论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Early Clin Dev Hematol Oncol & Cell Therapy, San Francisco, CA USA Bristol Myers Squibb, Oncogenesis ONC Themat Res Ctr TRC, San Francisco, CA USA
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Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaLu, Jun论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaYun, Weina论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaYang, Lingling论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaLou, Yude论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaSu, Dan论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaZhang, Shixuan论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaJin, Hanwei论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaLi, Xiang论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaSun, Jie论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaHuang, He论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaWang, Qishan论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Coll Anim Sci, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R ChinaJiang, Xi论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Bone Marrow Transplantat Ctr, Affiliated Hosp 1, Hangzhou, Peoples R China Zhejiang Univ, Inst Hematol, Hangzhou, Peoples R China Zhejiang Engn Lab Stem Cell & Immunotherapy, Hangzhou, Peoples R China Zhejiang Univ, Liangzhu Lab, Med Ctr, Hangzhou, Peoples R China Zhejiang Univ, Sch Med, Dept Pharmacol, Affiliated Hosp 1, Hangzhou, Peoples R China