Efficacy of poziotinib in HER2 exon 20 insertion NSCLC patients who received prior platinum-based and HER2 targeted therapies

被引:0
|
作者
Prelaj, A. [1 ]
Le, X. [2 ]
Proto, C. [3 ]
Baik, C. S. [4 ]
Tchekmedyian, N. [5 ]
Heymach, J. [6 ]
Bhat, G. [7 ]
Cornelissen, R. [8 ]
机构
[1] Fdn IRCCS Ist Nazl Tumori, Oncol Med Torac Dept, Milan, Italy
[2] Univ Texas MD Anderson Canc Ctr, Thorac Head & Neck, Houston, TX USA
[3] Fdn IRCCS Ist Nazl Tumori, Dept Med Oncol, Milan, Italy
[4] Univ Washington, Dept Med Oncol, Seattle Canc Care Alliance, Seattle, WA USA
[5] City Hope Natl Med Ctr, Med Oncol, Comprehens Canc Ctr, Duarte, CA USA
[6] MD Anderson Canc Ctr, Thorac Oncol, Houston, TX USA
[7] Spectrum Pharmaceut, Dept Clin Sci, Irvine, CA USA
[8] Erasmus MC Univ, Pulm Med, Med Ctr, Rotterdam, Netherlands
关键词
D O I
10.1016/j.annonc.2023.09.2422
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
1389P
引用
收藏
页数:1
相关论文
共 50 条
  • [21] Poziotinib administered twice daily improves safety and tolerability in patients with EGFR or HER2 exon 20 mutant NSCLC(ZENITH20-5).
    Le, Xiuning
    Shum, Elaine
    Suga, Jennifer M.
    Brahmer, Julie R.
    Dooms, Christophe
    Mamdani, Hirva
    Nechushtan, Hovav
    Riess, Jonathan W.
    Spira, Alexander
    Barrett, John A.
    Dreiling, Lyndah K.
    Socinski, Mark
    CANCER RESEARCH, 2021, 81 (13)
  • [22] Response Heterogeneity of EGFR and HER2 Exon 20 Insertions to Covalent EGFR and HER2 Inhibitors
    Kosaka, Takayuki
    Tanizaki, Junko
    Paranal, Raymond M.
    Endoh, Hideki
    Lydon, Christine
    Capelletti, Marzia
    Repellin, Claire E.
    Choi, Jihyun
    Ogino, Atsuko
    Calles, Antonio
    Ercan, Dalia
    Redig, Amanda J.
    Bahcall, Magda
    Oxnard, Geoffrey R.
    Eck, Michael J.
    Janne, Pasi A.
    CANCER RESEARCH, 2017, 77 (10) : 2712 - 2721
  • [23] Exploring optimal targeted combination therapies with neratinib for HER2 mutated NSCLC
    Kuraguchi, Mari
    Taus, Luke J.
    Zhou, Shan
    Avogadri-Connors, Francesca
    Cutler, Richard E.
    Lalani, Alshad S.
    Kirschmeier, Paul
    Janne, Pasi A.
    CANCER RESEARCH, 2018, 78 (13)
  • [24] HER2 protein quantification in multiple cancer indications identifies candidates for HER2 targeted therapies
    Sellappan, Shankar
    Schwartz, Sarit
    Wertheimer, Ellen
    Cecchi, Fabiola
    Mamus, Steven W.
    Catenacci, Daniel V. T.
    Hembrough, Todd
    CANCER RESEARCH, 2017, 77
  • [25] Case Series of HER2 Mutated Metastatic Lung Adenocarcinoma and Response to HER2 Targeted Therapies
    Chuang, Jody
    Neal, Joel W.
    Wakelee, Heather A.
    JOURNAL OF THORACIC ONCOLOGY, 2015, 10 (09) : S549 - S549
  • [26] Targeted therapy in NSCLC driven by HER2 insertions
    Peters, Solange
    Zimmermann, Stefan
    TRANSLATIONAL LUNG CANCER RESEARCH, 2014, 3 (02) : 84 - 88
  • [27] Discovery of potent, selective, and orally bioavailable HER2 tyrosine kinase inhibitors targeting HER2 exon20 insertion mutants and HER2WT
    Yoo, H. S.
    Jang, S. Y.
    Jeon, J.
    Nam, H. Y.
    Byun, J.
    Lee, G.
    Jeon, S.
    Chon, H.
    Kim, Y. Y.
    Park, H.
    An, Y. G.
    EUROPEAN JOURNAL OF CANCER, 2024, 211 : S44 - S45
  • [28] HER2 Targeted Therapies for Cancer and the Gastrointestinal Tract
    Al-Dasooqi, Noor
    Gibson, Rachel
    Bowen, Joanne
    Keefe, Dorothy
    CURRENT DRUG TARGETS, 2009, 10 (06) : 537 - 542
  • [29] Efficacy and safety of poziotinib in treatment-naive NSCLC harboring HER2 exon 20 mutations: A multinational phase II study (ZENITH20-4)
    Cornelissen, R.
    Sun, S.
    Wollner, M.
    Garassino, M. C. C.
    Prelaj, A.
    Haura, E. B.
    Piotrowska, Z.
    Goldman, J. W.
    Socinski, M.
    Dreling, L.
    Bhat, G.
    Lebel, F.
    Le, X.
    ANNALS OF ONCOLOGY, 2021, 32 : S1324 - S1324
  • [30] A Phase II Trial of Poziotinib in EGFR and HER2 exon 20 Mutant Non-Small Cell Lung Cancer (NSCLC)
    Heymach, J.
    Negrao, M.
    Robichaux, J.
    Carter, B.
    Patel, A.
    Altan, M.
    Gibbons, D.
    Fossella, F.
    Simon, G.
    Lam, V.
    Blumenschein, G.
    Tsao, A.
    Kurie, J.
    Mott, F.
    Jenkins, D.
    Mack, D.
    Feng, L.
    Roeck, B.
    Yang, Z.
    Papadimitrakopoulou, V.
    Elamin, Y.
    JOURNAL OF THORACIC ONCOLOGY, 2018, 13 (10) : S323 - S324