Application of the Knorr Reaction for the Directed Synthesis of Pyrazole Derivatives as Biologically Active Coligands for Gold Glyconanoparticles

被引:0
|
作者
Ershov, A. Y. [1 ]
Martynenkov, A. A. [1 ]
Lagoda, I. V. [2 ]
Batyrenko, A. A. [2 ]
机构
[1] Russian Acad Sci, Inst Macromol Cpds, St Petersburg 199004, Russia
[2] Minist Def Russian Federat, State Res Testing Inst Mil Med, St Petersburg 195043, Russia
关键词
thiolated hydrazide; Knorr reaction; pyrazoles; NANOPARTICLES;
D O I
10.1134/S1070428023110180
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The reaction of acetylacetone with 6-sulfanylhexanoic and 11-sulfanylundecanoic acid hydrazides was used to develop a method for the synthesis of previously unknown 1-(omega-sulfanylacyl)-3,5-dimethylpyrazoles as promising coligands for preparing gold glyconanoparticles for biomedical purposes.
引用
收藏
页码:1988 / 1989
页数:2
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