Synthesis of 14-epi-19-nor-22-oxa-1α,25-dihydroxyvitamin D3

被引:0
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作者
Wei Fan Li Hai Yong Wu Key Laboratory of Drag Targeting of Education Ministry
机构
关键词
1α; 25-Dihydroxyvitamin D3; 14-Epi-19-nor-22-oxa-1α; 25-dihydroxyvitamin D3; Device; Synthesis;
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中图分类号
O621.3 [有机合成化学];
学科分类号
070303 ; 081704 ;
摘要
The synthesis of 14-epi-19-nor-22-oxa-1α,25(OH);D;5 was started from diol 8 via Fall’s method,oxidation,epimerization, protection,coupling with the 19-nor-A-ring 7,and then deprotection of the hydroxyl functions.
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页码:259 / 260
页数:2
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