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- [31] Targeted protein degraders: a call for collective action to advance safety assessmentNATURE REVIEWS DRUG DISCOVERY, 2022, 21 (06) : 401 - 402Jones, Lyn H.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USA Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USAMitchell, Constance A.论文数: 0 引用数: 0 h-index: 0机构: Hlth & Environm Sci Inst, Washington, DC 17602 USA Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USALoberg, Lise论文数: 0 引用数: 0 h-index: 0机构: AbbVie, N Chicago, IL 60064 USA Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USAPavkovic, Mira论文数: 0 引用数: 0 h-index: 0机构: Bayer, Wuppertal, Germany Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USARao, Mohan论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Companies Johnson & Johnson, San Diego, CA USA Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USARoberts, Ruth论文数: 0 引用数: 0 h-index: 0机构: ApconiX, Alderley Edge, England Univ Birmingham, Dept Biosci, Birmingham, W Midlands, England Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USAStamp, Katie论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, New York, NY USA Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USAVolak, Laurie论文数: 0 引用数: 0 h-index: 0机构: Janssen Pharmaceut Companies Johnson & Johnson, San Diego, CA USA Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USAWittwer, Matthias B.论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche, Roche Innovat Ctr Basel, Basel, Switzerland Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USAPettit, Syril论文数: 0 引用数: 0 h-index: 0机构: Hlth & Environm Sci Inst, Washington, DC 17602 USA Dana Farber Canc Inst, Ctr Prot Degradat, Boston, MA 02115 USA
- [32] Biologics-based degraders - an expanding toolkit for targeted-protein degradationCURRENT OPINION IN BIOTECHNOLOGY, 2022, 78VanDyke, Derek论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USA Johns Hopkins Univ, Sch Med, Translat Tissue Engn Ctr, Baltimore, MD 21218 USA AstraZeneca, Biol Engn, R&D, Gaithersburg, MD USA Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USATaylor, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Biol Engn, R&D, Cambridge, England Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USAKaeo, Kyle J.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USA Johns Hopkins Univ, Sch Med, Translat Tissue Engn Ctr, Baltimore, MD 21218 USA Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USAHunt, James论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Biol Engn, R&D, Cambridge, England Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USASpangler, Jamie B.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USA Johns Hopkins Univ, Sch Med, Translat Tissue Engn Ctr, Baltimore, MD 21218 USA Johns Hopkins Univ, Bloomberg Kimmel Inst Canc Immunotherapy, Baltimore, MD 21218 USA Johns Hopkins Univ, Sidney Kimmel Comprehens Canc Ctr, Baltimore, MD 21218 USA Johns Hopkins Univ, Sch Med, Dept Biomed Engn, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Dept Oncol, Baltimore, MD 21205 USA Johns Hopkins Univ, Sch Med, Dept Ophthalmol, Baltimore, MD 21205 USA Johns Hopkins Univ, Dept Chem & Biomol Engn, Baltimore, MD 21218 USA
- [33] Development of natural product-based targeted protein degraders as anticancer agentsBIOORGANIC CHEMISTRY, 2024, 153Chen, Cheng论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaFeng, Yanyan论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaZhou, Chen论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Pharm, Dept Med Chem, Gainesville, FL 32610 USA Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaLiu, Zhouyan论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaTang, Ziwei论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaZhang, Ye论文数: 0 引用数: 0 h-index: 0机构: Changzhou Univ, Sch Petrochem Engn, Changzhou 213164, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaLi, Tong论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaGu, Chenglei论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R ChinaChen, Jichao论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China Nanjing Univ Chinese Med, Sch Pharm, Nanjing 210023, Peoples R China
- [34] Discovery of new targeted protein degraders using DNA-encoded chemistryCANCER RESEARCH, 2023, 83 (07)Keefe, Anthony D.论文数: 0 引用数: 0 h-index: 0Disch, Jeremy S.论文数: 0 引用数: 0 h-index: 0Duffy, Jennifer论文数: 0 引用数: 0 h-index: 0Lee, Esther C.论文数: 0 引用数: 0 h-index: 0Gikunju, Diana论文数: 0 引用数: 0 h-index: 0Chan, Betty论文数: 0 引用数: 0 h-index: 0Levin, Benjamin D.论文数: 0 引用数: 0 h-index: 0Monteiro, Michael I.论文数: 0 引用数: 0 h-index: 0Talcott, Sarah A.论文数: 0 引用数: 0 h-index: 0Lau, Anthony论文数: 0 引用数: 0 h-index: 0Zhou, Fei论文数: 0 引用数: 0 h-index: 0Kozhushnyan, Anton论文数: 0 引用数: 0 h-index: 0Westlund, Neil E.论文数: 0 引用数: 0 h-index: 0Mullins, Patrick B.论文数: 0 引用数: 0 h-index: 0Yu, Yan论文数: 0 引用数: 0 h-index: 0Von Rechenberg, Moritz论文数: 0 引用数: 0 h-index: 0Zhang, Junyi论文数: 0 引用数: 0 h-index: 0Arnautova, Yelena论文数: 0 引用数: 0 h-index: 0Liu, Yanbin论文数: 0 引用数: 0 h-index: 0Zhang, Ying论文数: 0 引用数: 0 h-index: 0McRiner, Andrew J.论文数: 0 引用数: 0 h-index: 0Kohlmann, Anna论文数: 0 引用数: 0 h-index: 0Clark, Matthew A.论文数: 0 引用数: 0 h-index: 0Cuozzo, John W.论文数: 0 引用数: 0 h-index: 0Huguet, Christelle论文数: 0 引用数: 0 h-index: 0Arora, Shilpi论文数: 0 引用数: 0 h-index: 0
- [35] Bifunctional Compounds as Molecular Degraders for Integrin- Facilitated Targeted Protein DegradationJOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 144 (48) : 21831 - 21836Zheng, Jiwei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaHe, Wanyi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China China Med Univ, Sch Pharm, Shenyang 110122, Liaoning, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaLi, Jing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China China Med Univ, Sch Pharm, Shenyang 110122, Liaoning, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaFeng, Xuejia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaLi, Yanyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaCheng, Binghua论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaZhou, Yimin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaLi, Meiqing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaLiu, Ke论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaShao, Ximing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaZhang, Jianchao论文数: 0 引用数: 0 h-index: 0机构: Southern Univ Sci & Technol, Sch Med, Dept Biochem, Shenzhen 518055, Guangdong, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaLi, Hongchang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaChen, Liang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R ChinaFang, Lijing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Chinese Acad Sci, Inst Biomed & Biotechnol, Shenzhen Inst Adv Technol, Shenzhen 518055, Guangdong, Peoples R China
- [36] Cure-PROs: Next-generation targeted protein degraders.JOURNAL OF CLINICAL ONCOLOGY, 2023, 41 (16)Giardina, Sarah F.论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USAValdambrini, Elena论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USAPeel, Michael论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USABacolod, Manny D.论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USARothenberg, Mace L.论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USALanman, Richard B.论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USAWarren, J. David论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USABarany, Francis论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med, New York, NY USA
- [37] Targeted protein degraders from an oncologist point of view: The Holy Grail of cancer therapy?CRITICAL REVIEWS IN ONCOLOGY HEMATOLOGY, 2022, 169Ambrosini, Margherita论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, ItalyFuca, Giovanni论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, ItalyDuca, Matteo论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, ItalyDamian, Silvia论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, ItalyDe Santis, Francesca论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, ItalyCorti, Francesca论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, ItalyCresta, Sara论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italyde Braud, Filippo论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Univ Milan, Oncol & Hematooncol Dept, Via Festa Perdono 7, I-20122 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, ItalyDi Nicola, Massimo论文数: 0 引用数: 0 h-index: 0机构: Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy Fdn IRCCS Ist Nazl Tumori, Med Oncol Dept, Via Venezian 1, I-20133 Milan, Italy
- [38] Simplifying Access to Targeted Protein Degraders via Nickel Electrocatalytic Cross-CouplingANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 63 (16)Neigenfind, Philipp论文数: 0 引用数: 0 h-index: 0机构: Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAMassaro, Luca论文数: 0 引用数: 0 h-index: 0机构: Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USA KTH Royal Inst Technol, Dept Chem, Teknikringen 30, S-10044 Stockholm, Sweden Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAPeter, Aron论文数: 0 引用数: 0 h-index: 0机构: Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USADegnan, Andrew P.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Early Dev, Small Mol Drug Discovery, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAEmmanuel, Megan A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, united States, Chem Proc Dev, 1 Squibb Dr, New Brunswick, NJ 08901 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAOderinde, Martins S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Early Dev, Small Mol Drug Discovery, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAHe, Chi论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Early Dev, Small Mol Drug Discovery, 10300 Campus Point Dr, San Diego, CA 92121 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAPeters, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Early Dev, Small Mol Drug Discovery, 10300 Campus Point Dr, San Diego, CA 92121 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAEl-Hayek Ewing, Tamara论文数: 0 引用数: 0 h-index: 0机构: Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USAKawamata, Yu论文数: 0 引用数: 0 h-index: 0机构: Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USABaran, Phil S.论文数: 0 引用数: 0 h-index: 0机构: Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USA Scripps Res, Dept Chem, 10550 North Torrey Pines Rd, La Jolla, CA 92037 USA
- [39] PK/PD modeling of targeted protein degraders: Charting new waters and navigating the shallowsDRUG DISCOVERY TODAY, 2025, 30 (03)Haid, Robin T. U.论文数: 0 引用数: 0 h-index: 0机构: Swiss Fed Inst Technol, Inst Pharmaceut Sci, Dept Chem & Appl Biosci, Zurich, Switzerland Bayer AG, Preclin Modeling & Simulat, Preclin Dev, Berlin, Germany Swiss Fed Inst Technol, Inst Pharmaceut Sci, Dept Chem & Appl Biosci, Zurich, SwitzerlandReichel, Andreas论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Preclin Modeling & Simulat, Preclin Dev, Berlin, Germany Swiss Fed Inst Technol, Inst Pharmaceut Sci, Dept Chem & Appl Biosci, Zurich, Switzerland
- [40] Targeted degraders clear first safety hurdlesNature Reviews Drug Discovery, 2020, 19 (7) : 435 - 435Asher Mullard论文数: 0 引用数: 0 h-index: 0