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- [42] New method for synthesis of EZH2 methyltransferase inhibitor GSK126SYNTHETIC COMMUNICATIONS, 2016, 46 (14) : 1215 - 1222Lu, Chen论文数: 0 引用数: 0 h-index: 0机构: Changzhou Univ, Sch Pharmaceut Engn & Life Sci, Changzhou 213164, Jiangsu, Peoples R China Changzhou Univ, Sch Pharmaceut Engn & Life Sci, Changzhou 213164, Jiangsu, Peoples R ChinaZhang, Qiang论文数: 0 引用数: 0 h-index: 0机构: Changzhou Univ, Sch Pharmaceut Engn & Life Sci, Changzhou 213164, Jiangsu, Peoples R China Changzhou Univ, Sch Pharmaceut Engn & Life Sci, Changzhou 213164, Jiangsu, Peoples R ChinaChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Changzhou Univ, Sch Pharmaceut Engn & Life Sci, Changzhou 213164, Jiangsu, Peoples R China Changzhou Univ, Sch Pharmaceut Engn & Life Sci, Changzhou 213164, Jiangsu, Peoples R China
- [43] EZH2 PARlyation is involved in PARP inhibitor sensitivity in breast cancer cellsCANCER SCIENCE, 2018, 109 : 559 - 559Yamaguchi, Hirohito论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USA
- [44] Design and Characterization of a Pyridone-Containing EZH2 Inhibitor Phosphate ProdrugJOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (03) : 1725 - 1732Kung, Pei-Pei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USAFan, Connie论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USAGukasyan, Hovhannes J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Pharmaceut Sci Res Enabling Grp, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USAHuang, Buwen论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USAKephart, Susan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USAKraus, Manfred论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USALee, Joseph H.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USASutton, Scott C.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USAYamazaki, Shinji论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Pharmacokinet Dynam & Metab, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USAZehnder, Luke论文数: 0 引用数: 0 h-index: 0机构: Pfizer Global Res & Dev, La Jolla Labs, Oncol Chem, San Diego, CA 92121 USA Pfizer Global Res & Dev, Oncol Res Unit, La Jolla Labs, San Diego, CA 92121 USA
- [45] PRECLINICAL CHARACTERIZATION OF E7438, A POTENT, SELECTIVE EZH2 INHIBITOR WITH ROBUST ANTITUMOR ACTIVITY AGAINST EZH2 MUTATED NHL XENOGRAFTS IN MICEANNALS OF ONCOLOGY, 2013, 24 : 13 - 13Keilhack, H.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USA
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New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USABunting, Karen L.论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USARosen, Monica论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAShen, Hao论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAYang, Shao Ning论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAWang, Ling论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAEzponda, Teresa论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Div Hematol Oncol, Robert H Lurie Comprehens Canc Ctr, Feinberg Sch Med, Chicago, IL 60611 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAMartinez-Garcia, Eva论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Div Hematol Oncol, Robert H Lurie Comprehens Canc Ctr, Feinberg Sch Med, Chicago, IL 60611 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAZhang, Haikuo论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAZheng, Yupeng论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Chem Life Proc Inst, Dept Chem, Evanston, IL 60208 USA Northwestern Univ, Chem Life Proc Inst, Dept Mol Biosci, Evanston, IL 60208 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAVerma, Sharad K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAMcCabe, Michael T.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAOtt, Heidi M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAVan Aller, Glenn S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAKruger, Ryan G.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USALiu, Yan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAMcHugh, Charles F.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAScott, David W.论文数: 0 引用数: 0 h-index: 0机构: British Columbia Canc Res Ctr, British Columbia Canc Agcy, Ctr Lymphoid Canc, Dept Pathol, Vancouver, BC V5Z 1L3, Canada British Columbia Canc Res Ctr, British Columbia Canc Agcy, Ctr Lymphoid Canc, Dept Expt Therapeut, Vancouver, BC V5Z 1L3, Canada Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAChung, Young Rock论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Dept Med, Leukemia Serv, New York, NY 10065 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAKelleher, Neil论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Chem Life Proc Inst, Dept Chem, Evanston, IL 60208 USA Northwestern Univ, Chem Life Proc Inst, Dept Mol Biosci, Evanston, IL 60208 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAShaknovich, Rita论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USACreasy, Caretha L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Oncol R&D, Canc Res, Canc Epigenet Discovery Performance Unit, Collegeville, PA 19426 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAGascoyne, Randy D.论文数: 0 引用数: 0 h-index: 0机构: British Columbia Canc Res Ctr, British Columbia Canc Agcy, Ctr Lymphoid Canc, Dept Pathol, Vancouver, BC V5Z 1L3, Canada British Columbia Canc Res Ctr, British Columbia Canc Agcy, Ctr Lymphoid Canc, Dept Expt Therapeut, Vancouver, BC V5Z 1L3, Canada Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAWong, Kwok-Kin论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USACerchietti, Leandro论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Dept Pharmacol, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USALevine, Ross L.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Dept Med, Leukemia Serv, New York, NY 10065 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAAbdel-Wahab, Omar论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Dept Med, Leukemia Serv, New York, NY 10065 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USALicht, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Div Hematol Oncol, Robert H Lurie Comprehens Canc Ctr, Feinberg Sch Med, Chicago, IL 60611 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAElemento, Olivier论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Inst Computat Biomed, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USAMelnick, Ari M.论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA Weill Cornell Med Coll, Dept Pharmacol, New York, NY 10021 USA Weill Cornell Med Coll, Div Hematol Oncol, Dept Med, New York, NY 10021 USA
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