Atomic structure of the trypsin-cyclotheonamide a complex. Lessons for the design of serine protease inhibitors

被引:0
|
作者
Lee, A.Y.
Hagihara, M.
Karmacharya, R.
Albers, M.W.
Schreiber, S.L.
Clardy, J.
机构
来源
| 1600年 / 115期
关键词
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
相关论文
共 50 条
  • [21] Predicted three-dimensional structural models of venom serine protease inhibitors and their interactions with trypsin and chymotrypsin
    Azim, MK
    Grossmann, JG
    Zaidi, ZH
    JOURNAL OF NATURAL TOXINS, 1999, 8 (03) : 363 - 384
  • [22] Atomic resolution crystal structure of HV-BBI protease inhibitor from amphibian skin in complex with bovine trypsin
    Grudnik, Przemyslaw
    Debowski, Dawid
    Legowska, Anna
    Malicki, Stanislaw
    Golik, Przemyslaw
    Karna, Natalia
    Rolka, Krzysztof
    Dubin, Grzegorz
    PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS, 2015, 83 (03) : 582 - 589
  • [23] Functional analysis of exosites 1 and 2 of thrombin in complex with serine protease inhibitors
    Fredenburgh, JC
    Stafford, AR
    Weitz, JI
    THROMBOSIS AND HAEMOSTASIS, 1999, : 698 - 698
  • [24] Structure-activity studies of cyclic ketone inhibitors of the serine protease plasmin: Design, synthesis, and biological activity
    Xue, Fengtian
    Seto, Christopher T.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2006, 14 (24) : 8467 - 8487
  • [25] Changes of trypsin in activity and secondary structure induced by complex with trypsin inhibitors and tea polyphenol
    Huang, Huihua
    Zhao, Mouming
    EUROPEAN FOOD RESEARCH AND TECHNOLOGY, 2008, 227 (02) : 361 - 365
  • [26] Changes of trypsin in activity and secondary structure induced by complex with trypsin inhibitors and tea polyphenol
    Huihua Huang
    Mouming Zhao
    European Food Research and Technology, 2008, 227 : 361 - 365
  • [27] Design and synthesis of novel and potent inhibitors of the type II transmembrane serine protease, matriptase, based upon the sunflower trypsin inhibitor-1
    Li, Peng
    Jiang, Sheng
    Lee, Sheau-Ling
    Lin, Cheng Yong
    Johnson, Michael D.
    Dickson, Robert B.
    Michejda, Christopher J.
    Roller, Peter P.
    JOURNAL OF MEDICINAL CHEMISTRY, 2007, 50 (24) : 5976 - 5983
  • [28] Structure-function relationships in serine protease-bovine pancreatic trypsin inhibitor interaction
    Krowarsch, D
    Zakrzewska, M
    Smalas, AO
    Otlewski, J
    PROTEIN AND PEPTIDE LETTERS, 2005, 12 (05): : 403 - 407
  • [29] Crystal structure of bovine duodenase, a serine protease, with dual trypsin and chymotrypsin-like specificities
    Pletnev, VZ
    Zamolodchikova, TS
    Pangborn, WA
    Duax, WL
    PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS, 2000, 41 (01) : 8 - 16
  • [30] Structure-based design of serine protease inhibitors:: Discovery of selective chymase inhibitors containing a novel β-amidophosphonic acid recognition motif
    Hawkins, MJ
    Greco, MN
    Powell, ET
    Corcoran, TW
    De Garavilla, L
    Kauffman, JA
    Wang, Y
    Minor, L
    Di Cera, E
    Sukumar, N
    Chen, ZW
    Pineda, AO
    Mathews, FS
    Maryanoff, BE
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U2693 - U2693