Selective N-methylation of ethyl esters of 3-(1H-imidazol-4-yl)-2-propenoic acid

被引：0
|
作者：
Mawlawi, H. [1 ]
Monje, M.C. [1 ]
Lattes, A. [1 ]
Rivière, M. [1 ]
机构：
[1] Laboratoire des IMRCP, URA Au CNRS 470, Université Paul Sabatier, 118 route de Narbonne, Toulouse Cédex,31062, France
来源：
Mathematical Problems in Engineering | 1992年 / 29卷 / 06期
关键词：
Methylation; -; Nitrogen; Esters;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Methods of selective methylation of the nitrogen atoms of the ethyl ester of 3-(1H-imidazol-4-yl)-2-pro-penoic acid are reported. The nitrogen atom α to the ethylenic chain was methylated after protection of the β nitrogen with a phenacyl group.
引用
收藏
页码：1621 / 1624
相关论文
共 50 条
  • [21] Bis[2-hydroxy-3-(1H-imidazol-4-yl)propionato]-nickel(II)
    Odoko, M
    Adachi, Y
    Okabe, N
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2002, 58 : M7 - M9
  • [22] PREPARATION AND CHARACTERIZATION OF S-[2-CARBOXY-1-(1H-IMIDAZOL-4-YL)ETHYL]GLUTATHIONE AND ITS DERIVATIVES AS PROPOSED PRECURSORS OF S-[2-CARBOXY-1-(1H-IMIDAZOL-4-YL)ETHYL]CYSTEINE, A COMPOUND FOUND IN HUMAN URINE
    KINUTA, M
    UBUKA, T
    YAO, K
    YAMADA, S
    YUKIHIRO, K
    TOMOZAWA, M
    BIOCHIMICA ET BIOPHYSICA ACTA, 1993, 1157 (02) : 192 - 198
  • [23] Bis[2-hydroxy-3-(1H-imidazol-4-yl)-propionato]cobalt(II)
    Okabe, N
    Adachi, Y
    ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 1999, 55 : 302 - 304
  • [24] Crystal structure of 2-(1H-imidazol-4-yl)-ethanaminium chloride
    Belfilali, Merle
    Yebdri, Siham
    Louhibi, Samira
    Boukli-hacene, Leila
    Roisnel, Thierry
    ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2015, 71 : O301 - U362
  • [25] SYNTHESIS AND CONNECTIVITY ASSIGNMENT (BY 2D-NMR) OF A NUCLEOSIDE-DIPEPTIDE - 5-[3-[[2-[[2-[[[2-AMINO]-1-OXO-3-[1H-IMIDAZOL-4-YL]PROPYL]AMINO]-1-OXO-3-[1H-IMIDAZOL-4-YL]PROPYL]AMINO]ETHYL]AMINO]-3-OXOPROPYL]-2'-DEOXYURIDINE
    BASHKIN, JK
    SONDHI, SM
    SAMPATH, U
    DAVIGNON, DA
    MODAK, AS
    NEW JOURNAL OF CHEMISTRY, 1994, 18 (03) : 305 - 316
  • [26] ISOLATION OF S-[2-CARBOXY-1-(1H-IMIDAZOL-4-YL)ETHYL]CYSTEINE FROM HUMAN URINE
    KINUTA, M
    UBUKA, T
    YAO, K
    FUTANI, S
    FUJIWARA, M
    KUROZUMI, Y
    BIOCHEMICAL JOURNAL, 1992, 283 : 39 - 40
  • [27] PHARMACOLOGICAL STUDIES ON THE TXA2 SYNTHETASE INHIBITOR (E)-3-[P-(1H-IMIDAZOL-1-YLMETHYL)PHENYL]-2-PROPENOIC ACID (OKY-046)
    HIRAKU, S
    TANIGUCHI, K
    WAKITANI, K
    OMAWARI, N
    KIRA, H
    MIYAMOTO, T
    OKEGAWA, T
    KAWASAKI, A
    UJIIE, A
    JAPANESE JOURNAL OF PHARMACOLOGY, 1986, 41 (03): : 393 - 401
  • [28] Efficient, Stereoselective Approach to the Synthesis of 3-(1-Phenyl-2-(Z-styrylsulfonyl)-1H-imidazol-4-yl)-2H-chromen-2-ones
    Guravaiah, Nalajam
    Rao, Vedula Rajeswar
    SYNTHETIC COMMUNICATIONS, 2011, 41 (08) : 1167 - 1174
  • [29] 3-(4-HYDROXY PHENYL)-2-PROPENOIC ACID - A REPRODUCTIVE INHIBITOR IN MALE-RAT
    PAKRASHI, A
    KABIR, SN
    RAY, H
    CONTRACEPTION, 1981, 23 (06) : 677 - 686
  • [30] Inhibitory Kinetics of 3-(4-Hydroxyphenyl)-2-Propenoic Acid on Tyrosinase-Catalyzing Reaction
    Gong, Sheng-zhao
    Chen, Qing-sheng
    INTERNATIONAL CONFERENCE ON BIOLOGICAL, MEDICAL AND CHEMICAL ENGINEERING (BMCE 2013), 2013, : 207 - 211
12345