共 50 条
- [21] Syntheses and biological evaluation of 5-(piperidin-1-yl)-3-phenyl-pentylsulfones as CCR5 antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (13) : 3589 - 3593Shankaran, K论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADonnelly, KL论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAShah, SK论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACaldwell, CG论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChen, P论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAFinke, PE论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAOates, B论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMacCoss, M论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMills, SG论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADeMartino, JA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGould, SL论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMalkowitz, L论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASiciliano, SJ论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASpringer, MS论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAKwei, G论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACarella, A论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACarver, G论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADanzelsen, R论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHolmes, K论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAKessler, J论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALineberger, J论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMiller, MD论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAEmini, EA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASchleif, WA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [22] 1-Methyl-3-{4-[(4-(2-oxo-2,3-dihydro-1H-benzirnidazol-1-yl)piperidin-1-yl)benzyl]}-2-phenylindoleMOLBANK, 2018, (04)论文数: 引用数: h-index:机构:Savrimoutou, Solene论文数: 0 引用数: 0 h-index: 0机构: Univ Bordeaux, UFR Sci Pharmaceut, Lab ARNA, INSERM U1212,UMR CNRS 5320, 146 Rue Leo Saignat, F-33076 Bordeaux, France Univ Bordeaux, UFR Sci Pharmaceut, Lab ARNA, INSERM U1212,UMR CNRS 5320, 146 Rue Leo Saignat, F-33076 Bordeaux, FranceRubio, Sandra论文数: 0 引用数: 0 h-index: 0机构: Univ Bordeaux, UFR Sci Pharmaceut, Lab ARNA, INSERM U1212,UMR CNRS 5320, 146 Rue Leo Saignat, F-33076 Bordeaux, France Univ Bordeaux, UFR Sci Pharmaceut, Lab ARNA, INSERM U1212,UMR CNRS 5320, 146 Rue Leo Saignat, F-33076 Bordeaux, France论文数: 引用数: h-index:机构:
- [23] Synthesis, antifungal and cytotoxic activities of 2-aryl-3-((piperidin-1-yl)ethyl)thiazolidinonesEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 64 : 74 - 80Kunzler, Alice论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, BrazilNeuenfeldt, Patricia D.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, Brazildas Neves, Adriana M.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, BrazilPereira, Claudio M. P.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, BrazilMarques, Gabriela H.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, Inst Biol, UFPel, Lab Micol, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, BrazilNascente, Patricia S.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, Inst Biol, UFPel, Lab Micol, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, BrazilFernandes, Maureen H. V.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, Fac Vet, UFPel, Lab Virol & Imunol, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, BrazilHuebner, Silvia O.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, Fac Vet, UFPel, Lab Virol & Imunol, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, BrazilCunico, Wilson论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, Brazil Univ Fed Pelotas, CCQFA, Lab Quim Aplicada Bioativos LaQuiABio, BR-96010900 Pelotas, RS, Brazil
- [24] Synthesis and evaluation of CCR5 antagonists containing modified 4-(piperidin-1-yl)-2-phenyl-1-(phenylsulfonylamino)-butane.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 222 : U657 - U657Shah, SK论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChen, N论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGuthikonda, RN论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMills, SG论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMacCoss, M论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMalkowitz, L论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASpringer, MS论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGould, SL论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADeMartino, JA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACarella, A论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACarver, G论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHolmes, K论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASchleif, WA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADanzeisen, R论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHazuda, D论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAKessler, J论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALineberger, J论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMiller, M论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAEmini, EA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [25] Discovery of 1-(4-(5-(5-amino-6-(5-tert-butyl-1,3,4-oxadiazol-2-yl) pyrazin-2-yl)-1-ethyl-1,2,4-triazol-3-yl) piperidin-1-yl)-3-hydroxypropan-1-one (AZD8835): A potent and selective inhibitor of PI3Kα and PI3Kδ for the treatment of cancersBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (22) : 5155 - 5162Barlaam, Bernard论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceCosulich, Sabina论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceDelouvrie, Bebedicte论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceEllston, Rebecca论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceFitzek, Martina论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceGermain, Herve论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceGreen, Stephen论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceHancox, Urs论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceHarris, Craig S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceHudson, Kevin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceLambert-van der Brempt, Christine论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceLebraud, Honorine论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceMagnien, Franoise论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceLamorlette, Maryannick论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceLe Griffon, Antoine论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceMorgentin, Remy论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceOuvry, Gilles论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FrancePage, Ken论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FrancePasquet, Georges论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FrancePolanska, Urszula论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceRuston, Linette论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceSaleh, Twana论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceVautier, Michel论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, FranceWard, Lara论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Oncol iMed, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Ctr Rech, ZI La Pompelle, F-51689 Reims 2, France
- [26] Synthesis and in-silico studies of 4-(5-(2-(4-(5-aryl-1,2,4-thiadiazol-3-yl) phenyl)-1H-imidazol-4-yl)-1,3,4-thiadiazol-2-yl)pyridinesRESULTS IN CHEMISTRY, 2024, 7Kethireddy, Shashikala论文数: 0 引用数: 0 h-index: 0机构: Geethanjali Coll Engn & Technol, Keesara 501301, India Geethanjali Coll Engn & Technol, Keesara 501301, IndiaEppakayala, Laxminarayana论文数: 0 引用数: 0 h-index: 0机构: Sreenidhi Inst Sci & Technol Autonomous Yamnampet, Hyderabad 501301, India Geethanjali Coll Engn & Technol, Keesara 501301, IndiaSyeda, Asra Banu论文数: 0 引用数: 0 h-index: 0机构: Jazan Univ, Coll Sci, Dept Chem, Al Maarefah Rd, Jazan 45142, Saudi Arabia Geethanjali Coll Engn & Technol, Keesara 501301, India
- [27] Discovery of Clinical Candidate 1-(4-(3-(4-(1H-Benzo[d]imidazole-2-carbonyl)phenoxy)pyrazin-2-yl)piperidin-1-yl)ethanone (AMG 579), A Potent, Selective, and Efficacious Inhibitor of Phosphodiesterase 10A (PDE10A)JOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (15) : 6632 - 6641Hu, Essa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAChen, Ning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USABourbeau, Matthew P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAHarrington, Paul E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USABiswas, Kaustav论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAKunz, Roxanne K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAAndrews, Kristin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAChmait, Samer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USADavis, Carl论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAMa, Ji论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAShi, Jianxia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USALester-Zeiner, Dianna论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USADanao, Jean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAAble, Jessica论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USACueva, Madelyn论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USATalreja, Santosh论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAKornecook, Thomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAChen, Hang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAPorter, Amy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAHungate, Randall论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USATreanor, James论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAAllen, Jennifer R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA
- [28] 3-[5-Methyl-1-(4-methylphenyl)-1H-1,2,3-triazol-4-yl]-N-phenyl-5-[4-(piperidin-1-yl) phenyl]-4,5-dihydro-1H-pyrazole-1-carbothioamide dimethyl-formamide hemisolvateACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2012, 68 : O1985 - +Abdel-Wahab, Bakr F.论文数: 0 引用数: 0 h-index: 0机构: Natl Res Ctr, Appl Organ Chem Dept, Giza 12622, Egypt Natl Res Ctr, Appl Organ Chem Dept, Giza 12622, EgyptMohamed, Hanan A.论文数: 0 引用数: 0 h-index: 0机构: Natl Res Ctr, Appl Organ Chem Dept, Giza 12622, Egypt Natl Res Ctr, Appl Organ Chem Dept, Giza 12622, EgyptNg, Seik Weng论文数: 0 引用数: 0 h-index: 0机构: Univ Malaya, Dept Chem, Kuala Lumpur 50603, Malaysia King Abdulaziz Univ, Chem Dept, Fac Sci, Jeddah, Saudi Arabia Natl Res Ctr, Appl Organ Chem Dept, Giza 12622, EgyptTiekink, Edward R. T.论文数: 0 引用数: 0 h-index: 0机构: Univ Malaya, Dept Chem, Kuala Lumpur 50603, Malaysia Natl Res Ctr, Appl Organ Chem Dept, Giza 12622, Egypt
- [29] 2-ethoxyphenyl)[4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl]methanoneACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2007, 63 : O642 - O643Naveen, S.论文数: 0 引用数: 0 h-index: 0机构: Univ Mysore, Dept Studies Phys, Mysore 570006, Karnataka, IndiaBasappa论文数: 0 引用数: 0 h-index: 0机构: Univ Mysore, Dept Studies Phys, Mysore 570006, Karnataka, IndiaSridhar, M. A.论文数: 0 引用数: 0 h-index: 0机构: Univ Mysore, Dept Studies Phys, Mysore 570006, Karnataka, India Univ Mysore, Dept Studies Phys, Mysore 570006, Karnataka, IndiaPrasad, J. Shashidhara论文数: 0 引用数: 0 h-index: 0机构: Univ Mysore, Dept Studies Phys, Mysore 570006, Karnataka, IndiaRangappa, K. S.论文数: 0 引用数: 0 h-index: 0机构: Univ Mysore, Dept Studies Phys, Mysore 570006, Karnataka, India
- [30] Synthesis and biological activity of 5-aryl-4-(4-(5-methyl-1H-imidazol-4-yl)piperidin-1-yl)pyrimidine analogs as potent, highly selective, and orally bioavailable NHE-1 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (18) : 4796 - 4799Atwal, Karnail S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USAO'Neil, Steven V.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USAAhmad, Saleem论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USADoweyko, Lidia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USAKirby, Mark论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USADorso, Charles R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USAChandrasena, Gamini论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USAChen, Bang-Chi论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USAZhao, Rulin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USAZahler, Robert论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Dept Discovery Chem, Princeton, NJ 08543 USA