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- [31] LY2969822: Pharmacological Characterization of an Orally Bioavailable Prodrug for a Potent, Selective mGlu2/3 Receptor AgonistCURRENT NEUROPHARMACOLOGY, 2014, 12 : 40 - 40McKinzie, D. L.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAJohnson, B. J.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAKnitowski, K.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAShaw, D.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USARorick-Kehn, L.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAKatner, J.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAPerry, K.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USASwanson, S.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USACatlow, J.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAJohnson, M. P.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAPrieto, L.论文数: 0 引用数: 0 h-index: 0机构: Alcobendas, Madrid, Spain Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USABeadle, C.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USAMonn, J. A.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Res Labs, Indianapolis, IN 46285 USA
- [32] Discovery of TK-642 as a highly potent, selective, orally bioavailable pyrazolopyrazine-based allosteric SHP2 inhibitorACTA PHARMACEUTICA SINICA B, 2024, 14 (08) : 3624 - 3642Tang, Kai论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaWang, Shu论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaFeng, Siqi论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaYang, Xinyu论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaGuo, Yueyang论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaRen, Xiangli论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaBai, Linyue论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaYu, Bin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Coll Chem, Pingyuan Lab, State Key Lab Antiviral Drugs, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Inst Adv Biomed Sci, Tianjian Lab Adv Biomed Sci, Zhengzhou 450000, Peoples R China Nanjing Univ, State Key Lab Pharmaceut Biotechnol, Nanjing 210023, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLiu, Hong-Min论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaSong, Yihui论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Key Lab Adv Drug Preparat Technol, Minist Educ, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China
- [33] Discovery of potent, highly selective, and orally bioavailable pyridine carboxamide c-jun NH2-terminal kinase inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (15) : 4455 - 4458Zhao, Hongyu论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASerby, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAXin, Zhili论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASzczepankiewicz, Bruce G.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALiu, Mei论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKosogof, Christi论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALiu, Bo论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USANelson, Lissa T. J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJohnson, Eric F.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAWang, Sanyi论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAPederson, Terry论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAGum, Rebecca J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAClampit, Jill E.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAHaasch, Deanna L.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAAbad-Zapatero, Cele论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAFry, Elizabeth H.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USARondinone, Cristina论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USATrevillyan, James M.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASham, Hing L.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALiu, Gang论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
- [34] TAS-116, a Novel, Orally Bioavailable HSP90a/β Selective Inhibitor Demonstrates Highly Potent Antitumor Activity in Preclinical Models with a Favorable PK ProfileEUROPEAN JOURNAL OF CANCER, 2012, 48 : 89 - 89Ohkubo, S.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanMuraoka, H.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanHashimoto, A.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanIto, S.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanIto, K.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanShibata, Y.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanKanoh, A.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanKitade, M.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanYonekura, K.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, JapanUtsugi, T.论文数: 0 引用数: 0 h-index: 0机构: Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan Taiho Pharmaceut Co LTD, Tsukuba Res Ctr, Tsukuba, Ibaraki, Japan
- [35] A Highly Potent, Orally Bioavailable Pyrazole-Derived Cannabinoid CB2 Receptor- Selective Full Agonist for In Vivo StudiesACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, 2024, 7 (08) : 2424 - 2438Chicca, Andrea论文数: 0 引用数: 0 h-index: 0机构: Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandBatora, Daniel论文数: 0 引用数: 0 h-index: 0机构: Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, Switzerland Univ Bern, Grad Sch Cellular & Biomed Sci, CH-3012 Bern, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandUllmer, Christoph论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandCaruso, Antonello论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandGruner, Sabine论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandFingerle, Ju''rgen论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandHartung, Thomas论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandDegen, Roland论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandMueller, Matthias论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandGrether, Uwe论文数: 0 引用数: 0 h-index: 0机构: Roche Pharm Res & Early Dev, Roche Innovat Ctr Basel, Pharmaceut Sci, CH-4070 Basel, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandPacher, Pal论文数: 0 引用数: 0 h-index: 0机构: NIAAA, Lab Cardiovasc Physiol & Tissue Injury PP, NIH, Bethesda, MD 20892 USA Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, SwitzerlandGertsch, Jurg论文数: 0 引用数: 0 h-index: 0机构: Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, Switzerland Univ Bern, Inst Biochem & Mol Med, CH-3012 Bern, Switzerland
- [36] Discovery and Characterization of 2-Aminooxazolines as Highly Potent, Selective, and Orally Active TAAR1 AgonistsACS MEDICINAL CHEMISTRY LETTERS, 2016, 7 (02): : 192 - 197Galley, Guido论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandBeurier, Angelica论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandDecoret, Guillaume论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandGoergler, Annick论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandHutter, Roman论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandMohr, Susanne论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandPaehler, Axel论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandSchmid, Philipp论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandTuerck, Dietrich论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandUnger, Robert论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandZbinden, Katrin Groebke论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandHoener, Marius C.论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, SwitzerlandNorcross, Roger D.论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland F Hoffmann La Roche Ltd, Roche Innovat Ctr, Pharma Res & Early Dev, CH-4070 Basel, Switzerland
- [37] Protein kinase B/Akt antagonists as antitumor agents part 4: Syntheses of potent, highly selective and orally bioavailable Akt inhibitors with reduced toxicity.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U133 - U133Gong, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAGandhi, VB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USALi, T论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USALuo, Y论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAShi, Y论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USALiu, X论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAKlinghofer, V论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USABouska, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAOlson, A论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAShoemaker, A论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAStoll, VS论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USALubbers, NL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAPolakowski, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USABallaron, S论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USACampbell, TJ论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USADe Jong, R论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAOltersdorf, T论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USALi, Q论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USARosenberg, SH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAGiranda, V论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USAZhu, GD论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res, Abbott Pk, IL 60064 USA
- [38] Discovery of XL01126: A Potent, Fast, Cooperative, Selective, Orally Bioavailable, and Blood-Brain Barrier Penetrant PROTAC Degrader of Leucine-Rich Repeat Kinase 2JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 144 (37) : 16930 - 16952Liu, Xingui论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandKalogeropulou, Alexia F.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandDomingos, Sofia论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandMakukhin, Nikolai论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, Scotland AstraZeneca, QMB Innovat Ctr, Oncol R&D, Tumour Targeted Delivery, 42 New Rd, London E1 2AX, England Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandNirujogi, Raja S.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandSingh, Francois论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandShpiro, Natalia论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandSaalfrank, Anton论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandSammler, Esther论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandGanley, Ian G.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandMoreira, Rui论文数: 0 引用数: 0 h-index: 0机构: Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, P-1649003 Lisbon, Portugal Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandAlessi, Dario R.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Sch Life Sci, Med Res Council MRC, Prot Phosphorylat & Ubiquitylat Unit, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, ScotlandCiulli, Alessio论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, Scotland Univ Dundee, Ctr Targeted Prot Degradat, Sch Life Sci, Div Biol Chem & Drug Discovery, Dundee DD1 5EH, Scotland
- [39] Discovery and optimization of a novel series of N-arylamide oxadiazoles as potent, highly selective and orally bioavailable cannabinoid receptor 2 (CB2) agonistsJOURNAL OF MEDICINAL CHEMISTRY, 2008, 51 (16) : 5019 - 5034Cheng, Yuan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAAlbrech, Brian K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USABrown, James论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USABuchanan, John L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USABuckner, William H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USADiMauro, Erin F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAEmkey, Renee论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAFremeau, Robert T., Jr.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAHarrnange, Jean-Christophe论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAHoffman, Beth J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAHuang, Liyue论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAHuang, Ming论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USALee, Josie Han论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USALin, Fen-Fen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Prot Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAMartin, Matthew W.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USANguyen, Hung Q.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Prot Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAPatel, Vinod F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USATomlinson, Susan A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAWhite, Ryan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Cambridge, MA 02139 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAXia, Xiaoyang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USAHitchcock, Stephen A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Chem Res & Discovery, Thousand Oaks, CA 91320 USA
- [40] A highly selective, orally bioavailable, vascular endothelial growth factor receptor-2 tyrosine kinase inhibitor has potent activity in vitro and in vivoANGIOGENESIS, 2009, 12 (03) : 287 - 296LaMontagne, Kenneth R.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut Inc, Florham Pk, NJ USA Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USAButler, Jeannene论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USABorowski, Virna B.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USAFuentes-Pesquera, Angel R.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USABlevitt, Jonathan M.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Dept Immunol, La Jolla, CA USA Novartis Pharmaceut Inc, Florham Pk, NJ USAHuang, Shenlin论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USALi, Ronghua论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USAConnolly, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USAGreenberger, Lee M.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Canc Therapeut Res, Raritan, NJ USA Novartis Pharmaceut Inc, Florham Pk, NJ USA