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- [23] Discovery of Potent, Selective, and Orally Bioavailable Small-Molecule Inhibitors of CDK8 for the Treatment of CancerJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (08) : 5439 - 5452Li, Yangguang论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaLiu, Yingtao论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaWu, Jianping论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaLiu, Xiaosong论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaWang, Lin论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaWang, Ju论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaYu, Jiaojiao论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaQi, Hongyun论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaQin, Luoheng论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaDing, Xiao论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaRen, Feng论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R ChinaZhavoronkov, Alex论文数: 0 引用数: 0 h-index: 0机构: Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China Insil Med Shanghai Ltd, Shanghai 201203, Peoples R China
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Whitehead Inst Biomed Res, Cambridge, MA 02142 USA MIT, Dept Biol, Cambridge, MA 02139 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAFicarro, Scott B.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Univ, Dept Biol Chem & Mol Pharmacol, Sch Med, Boston, MA 02115 USA Dana Farber Canc Inst, Blais Prote Ctr, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USADastur, Anahita论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Ctr Canc, Dept Med, Charlestown, MA 02129 USA Harvard Univ, Sch Med, Charlestown, MA 02129 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAAmzallag, Arnaud论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Ctr Canc, Dept Med, Charlestown, MA 02129 USA Harvard Univ, Sch Med, Charlestown, MA 02129 USA Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USARamaswamy, Sridhar论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Ctr Canc, Dept Med, Charlestown, MA 02129 USA Harvard Univ, Sch Med, Charlestown, MA 02129 USA Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USATesar, Bethany论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Dana Farber Canc Inst, Dept Med Oncol, Sch Med, Boston, MA 02115 USA Harvard Univ, Brigham & Womens Hosp, Dept Med, Sch Med, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAJenkins, Catherine E.论文数: 0 引用数: 0 h-index: 0机构: British Columbia Canc Agcy, Terry Fox Lab, Vancouver, BC V5Z 1L3, Canada Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAHannett, Nancy M.论文数: 0 引用数: 0 h-index: 0机构: Whitehead Inst Biomed Res, Cambridge, MA 02142 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAMcMillin, Douglas论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Dana Farber Canc Inst, Dept Med Oncol, Sch Med, Boston, MA 02115 USA Harvard Univ, Brigham & Womens Hosp, Dept Med, Sch Med, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USASanda, Takaomi论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Dana Farber Canc Inst, Dept Pediat Oncol, Sch Med, Boston, MA 02215 USA Natl Univ Singapore, Canc Sci Inst Singapore, Singapore 117599, Singapore Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USASim, Taebo论文数: 0 引用数: 0 h-index: 0机构: Korea Inst Sci & Technol, Chem Kinom Res Ctr, Seoul 136791, South Korea KU KIST Grad Sch Converging Sci & Technol, Seoul 136713, South Korea Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAKim, Nam Doo论文数: 0 引用数: 0 h-index: 0机构: Daegu Gyeongbuk Med Innovat Fdn, Taegu 706010, South Korea Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USALook, Thomas论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Dana Farber Canc Inst, Dept Pediat Oncol, Sch Med, Boston, MA 02215 USA Childrens Hosp, Div Hematol Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAMitsiades, 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Biol, Boston, MA 02115 USA Harvard Univ, Dept Biol Chem & Mol Pharmacol, Sch Med, Boston, MA 02115 USA Dana Farber Canc Inst, Blais Prote Ctr, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAYoung, Richard A.论文数: 0 引用数: 0 h-index: 0机构: Whitehead Inst Biomed Res, Cambridge, MA 02142 USA MIT, Dept Biol, Cambridge, MA 02139 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Univ, Dept Biol Chem & Mol Pharmacol, Sch Med, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA
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