A CONVENIENT PREPARATION OF MONOSUBSTITUTED N,N'-DI(BOC)-PROTECTED GUANIDINES

被引：0

作者：

DRAKE, B ^{[1
]}

PATEK, M ^{[1
]}

LEBL, M ^{[1
]}

机构：

[1] SECECTIDE CORP,TUCSON,AZ 85737

来源：

SYNTHESIS-STUTTGART | 1994年 / 06期

关键词：

DI(BOC)-PROTECTED GUANIDINES; GUANYLATION; ARGININE ANALOGS;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1-H-Pyrazole-1-[N,N'-bis(tert-butoxycarbonyl)]carboxamidine (1) reacts under mild conditions with a number of amines and amino acids to give the respective protected guanidines in moderate to high isolated yields.

引用

页码：579 / 582

页数：4

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