A CONVENIENT PREPARATION OF MONOSUBSTITUTED N,N'-DI(BOC)-PROTECTED GUANIDINES

被引：0
|
作者：
DRAKE, B [1 ]
PATEK, M [1 ]
LEBL, M [1 ]
机构：
[1] SECECTIDE CORP,TUCSON,AZ 85737
来源：
SYNTHESIS-STUTTGART | 1994年 / 06期
关键词：
DI(BOC)-PROTECTED GUANIDINES; GUANYLATION; ARGININE ANALOGS;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
1-H-Pyrazole-1-[N,N'-bis(tert-butoxycarbonyl)]carboxamidine (1) reacts under mild conditions with a number of amines and amino acids to give the respective protected guanidines in moderate to high isolated yields.
引用
收藏
页码：579 / 582
页数：4
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