CHARACTERIZATION OF THE ATPASE ACTIVITY OF THE MR 170,000 TO 180,000 MEMBRANE GLYCOPROTEIN (P-GLYCOPROTEIN) ASSOCIATED WITH MULTIDRUG RESISTANCE IN K562/ADM CELLS

被引:0
|
作者
HAMADA, H [1 ]
TSURUO, T [1 ]
机构
[1] JAPANESE FDN CANC RES, CTR CANC CHEMOTHERAPY, KAMI IKEBUKURO, TOSHIMA KU, TOKYO 170, JAPAN
关键词
D O I
暂无
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:4926 / 4932
页数:7
相关论文
共 50 条
  • [41] Effect of Phorbol 12-Myristate 13-Acetate on Function and Gene Expression of P-Glycoprotein in Adriamycin-Resistant K562/ADM Cells
    Li, Yuhua
    Bi, Huichang
    Zhong, Guoping
    Huang, Ling
    Li, Gelin
    Xia, Yanzhe
    Chen, Xiao
    Huang, Min
    PHARMACOLOGY, 2013, 92 (3-4) : 121 - 130
  • [42] Osthole shows the potential to overcome P-glycoprotein-mediated multidrug resistance in human myelogenous leukemia K562/ADM cells by inhibiting the PI3K/Akt signaling pathway
    Wang, Hong
    Jia, Xiu-Hong
    Chen, Jie-Ru
    Wang, Jian-Yong
    Li, You-Jie
    ONCOLOGY REPORTS, 2016, 35 (06) : 3659 - 3668
  • [43] INHIBITION BY ERYTHROID-DIFFERENTIATION FACTOR (ACTIVIN-A) OF P-GLYCOPROTEIN EXPRESSION IN MULTIDRUG-RESISTANT HUMAN K562 ERYTHROLEUKEMIA-CELLS
    OKABEKADO, J
    HAYASHI, M
    HONMA, Y
    HOZUMI, M
    TSURUO, T
    CANCER RESEARCH, 1991, 51 (10) : 2582 - 2586
  • [44] Characterization of H+-ATPase-dependent activity of multidrug resistance-associated protein in homoharringtonine-resistant human leukemic K562 cells
    Z Benderra
    H Morjani
    A Trussardi
    M Manfait
    Leukemia, 1998, 12 : 1539 - 1544
  • [45] Reversal of P-glycoprotein-mediated multidrug resistance by guggulsterone in doxorubicin-resistant human myelogenous leukemia (K562/DOX) cells
    Xu, Hong-Bin
    Li, Ling
    Liu, Guo-Qing
    PHARMAZIE, 2009, 64 (10): : 660 - 665
  • [46] Modulation of P-glycoprotein activity by the substituted quinoxalinone compound QA3 in adriamycin-resistant K562/A02 cells
    Li-Rui Sun
    Julia Li Zhong
    Shu-Xiang Cui
    Xun Li
    Stephen Geoffrey Ward
    Yan-Qiu Shi
    Xiao-Fan Zhang
    Yan-Na Cheng
    Jian-Jun Gao
    Xian-Jun Qu
    Pharmacological Reports, 2010, 62 : 333 - 342
  • [47] Designed P-glycoprotein inhibitors with triazol-tetrahydroisoquinoline-core increase doxorubicin-induced mortality in multidrug resistant K562/A02 cells
    Kairuki, Mutta
    Qiu, Qianqian
    Pan, Miaobo
    Li, Qifei
    Zhou, Jiaqi
    Ghaleb, Hesham
    Huang, Wenlong
    Qian, Hai
    Jiang, Cheng
    BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 27 (15) : 3347 - 3357
  • [48] Modulation of P-glycoprotein activity by the substituted quinoxalinone compound QA3 in adriamycin-resistant K562/A02 cells
    Sun, Li-Rui
    Zhong, Julia Li
    Cui, Shu-Xiang
    Li, Xun
    Ward, Stephen Geoffrey
    Shi, Yan-Qiu
    Zhang, Xiao-Fan
    Cheng, Yan-Na
    Gao, Jian-Jun
    Qu, Xian-Jun
    PHARMACOLOGICAL REPORTS, 2010, 62 (02) : 333 - 342
  • [49] INVITRO BONE-MARROW PURGING OF MULTIDRUG-RESISTANT CELLS WITH A MOUSE MONOCLONAL-ANTIBODY DIRECTED AGAINST MR 170,000 GLYCOPROTEIN AND A SAPORIN-CONJUGATED ANTI-MOUSE ANTIBODY
    DINOTA, A
    TAZZARI, PL
    MICHIELI, M
    VISANI, G
    GOBBI, M
    BONTADINI, A
    TASSI, C
    FANIN, R
    DAMIANI, D
    GRANDI, M
    PILERI, S
    BOLOGNESI, A
    STIRPE, F
    BACCARANI, M
    TSURUO, T
    TURA, S
    CANCER RESEARCH, 1990, 50 (14) : 4291 - 4294
  • [50] Synthesis of New Steroidal Inhibitors of P-Glycoprotein-Mediated Multidrug Resistance and Biological Evaluation on K562/R7 Erythroleukemia Cells
    de Ravel, Marc Rolland
    Alameh, Ghina
    Melikian, Maxime
    Mahiout, Zahia
    Emptoz-Bonneton, Agnes
    Matera, Eva-Laure
    Lomberget, Thierry
    Barret, Roland
    Rocheblave, Luc
    Walchshofer, Nadia
    Beltran, Sonia
    El Jawad, Lucienne
    Mappus, Elisabeth
    Grenot, Catherine
    Pugeat, Michel
    Dumontet, Charles
    Le Borgne, Marc
    Cuilleron, Claude Yves
    JOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (04) : 1832 - 1845