BLOCKADE OF THE PLATELET TXA2 PGH2 RECEPTOR BY A PHOTOAFFINITY LIGAND

被引:0
|
作者
ZEHENDER, H
WITTE, EC
WOLFF, HP
STEGMEIER, K
PATSCHEKE, H
机构
[1] UNIV HEIDELBERG,KLINIKUM MANNHEIM,INST CLIN CHEM,D-6800 MANNHEIM,FED REP GER
[2] BOEHRINGER MANNHEIM GMBH,DEPT MED RES,D-6800 MANNHEIM,FED REP GER
关键词
D O I
暂无
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:64 / 64
页数:1
相关论文
共 50 条
  • [31] PGH2, TXA2 AND PGI2 HAVE POTENT AND DIFFERENTIATED ACTIONS ON HUMAN UTERINE CONTRACTILITY
    WILHELMSSON, L
    WIKLAND, M
    WIQVIST, N
    PROSTAGLANDINS, 1981, 21 (02): : 277 - 286
  • [32] PLATELET TXA2 SYNTHETASE INHIBITION AND TXA2 PROSTAGLANDIN ENDOPEROXIDE RECEPTOR BLOCKADE COMBINED IN ONE MOLECULE (R 68070)
    DECLERCK, F
    VANDEWIELE, R
    XHONNEUX, B
    VANGORP, L
    SOMERS, Y
    LOOTS, W
    BEETENS, J
    VANWAUWE, J
    FREYNE, E
    JANSSEN, PAJ
    THROMBOSIS AND HAEMOSTASIS, 1987, 58 (01) : 181 - 181
  • [33] PICOTAMIDE INHIBITS TXA2/PGH2 RECEPTORS OF MUSCLE VASCULAR CELLS FROM HUMAN ARTERIES
    MODESTI, PA
    COLELLA, A
    CECIONI, I
    COSTOLI, A
    SERNERI, GGN
    THROMBOSIS AND HAEMOSTASIS, 1993, 69 (06) : 669 - 669
  • [34] BINDING OF A THROMBOXANE A2 PROSTAGLANDIN-H2 (TXA2/PGH2) RECEPTOR ANTAGONIST TO WASHED HUMAN-PLATELETS
    MAIS, DE
    HALUSHKA, PV
    CIRCULATION, 1985, 72 (04) : A7 - A7
  • [35] PHARMACOLOGICAL PROPERTIES OF KT2-962, AN AZULENE DERIVATIVE, A NOVEL TXA2 PGH2 ANTAGONIST
    KOSAKAI, K
    WAKABAYASHI, S
    SATOH, T
    TOMIYAMA, A
    SATAKE, N
    SHIBATA, S
    FASEB JOURNAL, 1991, 5 (04): : A500 - A500
  • [36] Salt loading enhances rat renal TxA2/PGH2 receptor expression and TGF response to U-46,619
    Welch, WJ
    Peng, B
    Takeuchi, K
    Abe, K
    Wilcox, CS
    AMERICAN JOURNAL OF PHYSIOLOGY-RENAL PHYSIOLOGY, 1997, 273 (06) : F976 - F983
  • [37] The presence of the TXA2 receptor in lipid rafts of platelets is necessary for platelet activation by TXA2
    Moscardo, Antonio
    Valles, Juana
    Madrid, Isabel
    Latorre, Ana
    Dasi, Angeles
    Teresa Santos, Maria
    THROMBOSIS RESEARCH, 2012, 130 : S103 - S103
  • [38] PROSTACYCLIN (PGI2)- AND THROMBOXANE (TXA2/PGH2) RECEPTORS IN PLATELETS AND VESSEL WALL IN CONTROL CONDITIONS AND ISCHEMIA
    JASCHONEK, K
    HAEMOSTASIS, 1986, 16 : 43 - 43
  • [39] SYNTHESIS OF [17,18-H-3] TRANS-13-AZAPROSTANOIC ACID - A LABELED PROBE FOR THE PGH2/TXA2 RECEPTOR
    GHALI, NI
    KATTELMAN, EJ
    HUNG, SC
    SCHNORF, KE
    LEBRETON, GC
    VENTON, DL
    PROSTAGLANDINS, 1984, 27 (06): : 865 - 876
  • [40] SYNTHESES OF NEW TXA2/PGH2-RECEPTOR ANTAGONISTS AND THEIR BIOLOGICAL PROPERTIES
    DEICKE, P
    KLAR, U
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1992, 2 (09) : 1063 - 1068