Synthesis of Fused Heterocyclic Compounds Derived from 2-Phenyl[1,5] benzothiazepin-4(5H)-One

被引：0
|
作者：
Khodairy, A. [1 ]
Hassan, N. S. [1 ]
El-Wassimy, M. T. [1 ]
机构：
[1] Sohag Univ, Fac Sci, Chem Dept, Sohag, Egypt
来源：
EGYPTIAN JOURNAL OF CHEMISTRY | 2011年 / 54卷 / 03期
关键词：
1,5-Benzothiazepin-4(5H)-one; Naphthyridines and Thieno [3,2-e] benzothiazepines;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
2-PHENYL[1,5] benzothiazepin-4(5H)-one (1) was reacted with arylidenenitriles, a mixture of carbon disulphide or phenylisothiocyanate and active nitriles to give pyrano-, pyrido-, thiopyrano-, 1,2dithiolo[ 3,4-e]-; 1,3-dithiolo[4,5-e] [1,5] benzothiazepines, benzothiazepino-[ 6,5-c] [1,8] naphthyridine and oxathieno [1, 5] benzothiazepines (2-11), respectively. Treatment of compound 1 with a mixture of sulphur and phenyl isothiocyanate or 2-amino-1,1,3-tricyano-2aminopropene gave 1,3-dithieno [4,5-e]-and thieno [3,2-e]-[1,5] benzothiazepines (12, 13), respectively.
引用
收藏
页码：349 / 359
页数：11
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