ENZYMATIC REGIOSELECTIVE ACYLATION OF THE 3'-HYDROXYL GROUPS OF 2'-DEOXY-5-FLUOROURIDINE (FUDR) AND 2'-DEOXY-5-TRIFLUOROMETHYLURIDINE (CF3UDR)

被引：23
|
作者：
NOZAKI, K
UEMURA, A
YAMASHITA, J
YASUMOTO, M
机构：
[1] Chemical Synthesis Research Laboratory, Taiho Pharmaceutical Co., Ltd., Kodama-gun, Saitama
来源：
TETRAHEDRON LETTERS | 1990年 / 31卷 / 50期
关键词：
D O I：
10.1016/S0040-4039(00)88556-1
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A lipase from Pseudomonas sp. (Amano PS) catalyzes regioselecfive acylation of the 3′-hydroxyl groups of FUdR and CF3UdR. © 1990.
引用
收藏
页码：7327 / 7328
页数：2
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