IS THE SELECTIVE NONPEPTIDE NK-1 RECEPTOR ANTAGONIST CP96,345 A PERIPHERALLY ACTING ANALGESIC

被引:8
|
作者
BERGE, OG
STAHLBERG, M
机构
[1] Astra Pain Control, Preclinical Research, Södertälje
关键词
SUBSTANCE-P; CP96,345; PAIN; ANALGESIA; NOCICEPTION; NK-1; INFLAMMATION;
D O I
10.1016/0167-0115(93)90110-T
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
[No abstract available]
引用
收藏
页码:430 / 432
页数:3
相关论文
共 50 条
  • [31] THE EFFECT OF VAGAL COOLING, VAGOTOMY AND THE NK-1 ANTAGONIST-CP-96,345 ON THE BRONCHOMOTOR RESPONSE TO SUBSTANCE-P IN NORMAL SHEEP
    CORCORAN, BM
    HAIGH, AL
    REGULATORY PEPTIDES, 1992, 39 (2-3) : 271 - 271
  • [32] INTERACTION OF THE NONPEPTIDE NK1 TACHYKININ RECEPTOR ANTAGONIST (+/-)CP-96,345 WITH L-TYPE CALCIUM CHANNELS IN RAT CEREBRAL-CORTEX
    GUARD, S
    WATLING, KJ
    BRITISH JOURNAL OF PHARMACOLOGY, 1992, 106 : P37 - P37
  • [33] PREPARATION AND RADIOLABELING OF CP-96,345, THE 1ST NONPEPTIDE SUBSTANCE-P ANTAGONIST
    LOWE, JA
    DROZDA, SE
    SNIDER, RM
    LONGO, KP
    BORDNER, J
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1991, 1 (02) : 129 - 132
  • [34] STEREOSPECIFIC EFFECTS OF A NONPEPTIDIC NK1 SELECTIVE ANTAGONIST, CP-96,345 - ANTINOCICEPTION IN THE ABSENCE OF MOTOR DYSFUNCTION
    YAMAMOTO, T
    YAKSH, TL
    LIFE SCIENCES, 1991, 49 (26) : 1955 - 1963
  • [35] Photoaffinity labeling of the substance P (NK-1) receptor by [H-3(2)]-azido-CP-96,345, a photoreactive derivative of a non-peptide antagonist.
    Macdonald, D
    Silberman, SC
    Leeman, SE
    Boyd, ND
    FASEB JOURNAL, 1996, 10 (03): : 3958 - 3958
  • [36] NK-1, BUT NOT NK-2, TACHYKININ RECEPTORS MEDIATE PLASMA EXTRAVASATION INDUCED BY ANTIDROMIC C-FIBER STIMULATION IN RAT HINDPAW - DEMONSTRATED WITH THE NK-1 ANTAGONIST CP-96,345 AND THE NK-2 ANTAGONIST MEN-10207
    XU, XJ
    DALSGAARD, CJ
    MAGGI, CA
    WIESENFELDHALLIN, Z
    NEUROSCIENCE LETTERS, 1992, 139 (02) : 249 - 252
  • [37] THE INTERACTION OF THE NK(1) RECEPTOR ANTAGONIST CP-96,345 WITH L-TYPE CALCIUM CHANNELS AND ITS FUNCTIONAL CONSEQUENCES
    GUARD, S
    BOYLE, SJ
    TANG, KW
    WATLING, KJ
    MCKNIGHT, AT
    WOODRUFF, GN
    BRITISH JOURNAL OF PHARMACOLOGY, 1993, 110 (01) : 385 - 391
  • [38] CP-99,994, A NONPEPTIDE ANTAGONIST OF THE TACHYKININ NK(1) RECEPTOR
    MCLEAN, S
    SNIDER, RM
    DESAI, MC
    ROSEN, T
    BRYCE, DK
    LONGO, KP
    SCHMIDT, AW
    HEYM, J
    REGULATORY PEPTIDES, 1993, 46 (1-2) : 329 - 331
  • [39] NONPEPTIDE ANTAGONISTS, CP-96,345 AND RP-67580, DISTINGUISH SPECIES VARIANTS IN TACHYKININ NK(1)-RECEPTORS
    BARR, AJ
    WATSON, SP
    BRITISH JOURNAL OF PHARMACOLOGY, 1993, 108 (01) : 223 - 227
  • [40] ROLE OF NK1 TACHYKININ RECEPTORS IN THERMONOCICEPTION - EFFECT OF (+/-)-CP 96,345, A NONPEPTIDE SUBSTANCE-P ANTAGONIST, ON THE HOT PLATE TEST IN MICE
    LECCI, A
    GIULIANI, S
    PATACCHINI, R
    VITI, G
    MAGGI, CA
    NEUROSCIENCE LETTERS, 1991, 129 (02) : 299 - 302