PREPARATION OF N-ARYLATED HETEROCYCLES BY NUCLEOPHILIC AROMATIC-SUBSTITUTION

被引：48
|
作者：
STABLER, SR
JAHANGIR
机构：
[1] Institute of Organic Chemistry, Syntex Discovery Research, Palo Alto
来源：
SYNTHETIC COMMUNICATIONS | 1994年 / 24卷 / 01期
关键词：
D O I：
10.1080/00397919408012635
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Nucleophilic aromatic substitution of fluorobenzoates and fluorophenylnitriles with weakly basic heterocycles readily occur. This synthetic methodology is utillized to produce potent angiotensin-II antagonists.
引用
收藏
页码：123 / 129
页数：7
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