REACTION OF 1-AMINOPHTHALAZINES WITH ALPHA-HALOCARBONYL COMPOUNDS - IMIDAZO[2,1-A]PHTHALAZINES AND THEIR BENZODIAZEPINE RECEPTOR ACTIVITIES

被引：0
|
作者：
CATARZI, D
CECCHI, L
COLOTTA, V
CONTI, G
MELANI, F
FILACCHIONI, G
MARTINI, C
GIUSTI, L
LUCACCHINI, A
机构：
[1] UNIV FLORENCE,DIPARTIMENTO SCI FARMACEUT,VIA GINO CAPPONI 9,I-50121 FLORENCE,ITALY
[2] UNIV PISA,IST POLICATTEDRA DISCIPLINE BIOL,I-56100 PISA,ITALY
来源：
FARMACO | 1993年 / 48卷 / 04期
关键词：
D O I：
暂无
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
The one-pot synthesis and the benzodiazepine receptor binding activity of some imidazo[2,1-a]phthalazines bearing different substituents at position-2 and/or 3 and/or 6 is reported. The dissimilar binding results of the reported compounds are discussed in relation to the nature and/or position of the substituents on the tricyclic ring system.
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页码：447 / 457
页数：11
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