STUDIES ABOUT THE CYCLIZATION OF 1,2-DIAMINES WITH ALDEHYDES AND KETONES

被引：0
|
作者：
LESSEL, J
机构：
来源：
PHARMAZIE | 1994年 / 49卷 / 09期
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D O I：
暂无
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
The reaction of the 1,2-dinucleophile ethylendiamine with benzaldehydes yields diimines, from o-phenylendiamine monoimines respectively benzimidazoles are formed. beta-Diketones give 1,5-benzodiazepines. The different behaviour is explained by MNDO calculations and by perturbation theory.
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页码：649 / 653
页数：5
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