STRUCTURAL REQUIREMENTS FOR AGONIST ACTIONS OF BETA-CARBOLINES AT THE BENZODIAZEPINE RECEPTOR (BZR) - ALIGNMENT RULE AND PHARMACOPHORE FOR FULL AND PARTIAL AGONISTS AT THE BZR

被引：0

作者：

DIAZARAUZO, H ^{[1
]}

SKOLNICK, P ^{[1
]}

COOK, JM ^{[1
]}

机构：

[1] UNIV WISCONSIN,DEPT CHEM,MILWAUKEE,WI 53201

来源：

ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 1990年 / 200卷

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：45 / MEDI

共 12 条

[1] THE USE OF BETA-CARBOLINES TO FURTHER DIFFERENTIATE THE AGONIST INVERSE AGONIST PHARMACOPHORE AT THE BZR
COX, ED
COOK, JM
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1994, 208 : 192 - MEDI
[2] BENZODIAZEPINE-RECEPTOR (BZR) LIGANDS - THE CONFORMATIONAL FIT OF AGONIST-BETA-CARBOLINES TO AN IMIDAZOBENZODIAZEPINE TEMPLATE
FRYER, RI
WANG, CG
CHIA, NC
BASILE, AS
GU, ZQ
SKOLNICK, P
MEDICINAL CHEMISTRY RESEARCH, 1995, 5 (04) : 296 - 307
[3] BENZODIAZEPINE RECEPTOR LIGAND ACTIONS ON GABA RESPONSES - BETA-CARBOLINES, PURINES
SKERRITT, JH
MACDONALD, RL
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 101 (1-2) : 135 - 141
[4] SYNTHESIS OF NOVEL 3-SUBSTITUTED BETA-CARBOLINES AS BENZODIAZEPINE RECEPTOR LIGANDS - PROBING THE BENZODIAZEPINE RECEPTOR PHARMACOPHORE
ALLEN, MS
HAGEN, TJ
TRUDELL, ML
CODDING, PW
SKOLNICK, P
COOK, JM
JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (09) : 1854 - 1861
[5] DISCRIMINATIVE STIMULUS PROPERTIES OF THE BENZODIAZEPINE RECEPTOR PARTIAL AGONIST BETA-CARBOLINES ABECARNIL AND ZK 95962 - A COMPARISON WITH CHLORIAZEPOXIDE
ANDREWS, JS
STEPHENS, DN
BEHAVIOURAL PHARMACOLOGY, 1991, 2 (03): : 171 - 185
[6] SYNTHESIS OF 6-SUBSTITUTED BETA-CARBOLINES THAT BEHAVE AS BENZODIAZEPINE RECEPTOR ANTAGONISTS OR INVERSE AGONISTS
HAGEN, TJ
SKOLNICK, P
COOK, JM
JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (04) : 750 - 753
[7] BETA-CARBOLINES CHARACTERIZED AS BENZODIAZEPINE RECEPTOR AGONISTS AND INVERSE AGONISTS PRODUCE BIDIRECTIONAL CHANGES IN PALATABLE FOOD-CONSUMPTION
COOPER, SJ
BRAIN RESEARCH BULLETIN, 1986, 17 (05) : 627 - 637
[8] SYNTHESIS OF 6-SUBSTITUTED BETA-CARBOLINES WHICH BEHAVE AS BENZODIAZEPINE RECEPTOR ANTAGONISTS OR INVERSE AGONISTS
HAGEN, TJ
SKOLNICK, P
COOK, JM
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1987, 193 : 35 - MEDI
[9] EFFECT ON HYPOTHALAMIC SELF-STIMULATION OF THE NOVEL BETA-CARBOLINES ZK-93-426 (A BENZODIAZEPINE RECEPTOR ANTAGONIST) AND ZK-91-296 (A PUTATIVE PARTIAL AGONIST)
HERBERG, LJ
MONTGOMERY, AMJ
FILE, SE
PELLOW, S
STEPHENS, DN
JOURNAL OF NEURAL TRANSMISSION, 1986, 66 (02) : 75 - 84
[10] Studies of the pharmacophore/receptor models for benzodiazepine receptor subtypes. Binding affinities of substituted beta-carbolines for alpha chi beta 3 gamma 2 (x=1, 2, 3, 5, or 6) subtypes and a comparative molecular field analysis.
Huang, Q
Cox, ED
Gan, T
Bennett, DW
Cook, JM
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 212 : 157 - MEDI

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