ABSORPTION AND BIOAVAILABILITY EVALUATION OF ORALLY ACTIVE RENIN INHIBITOR ABBOTT-72517 IN THE DOG

被引:0
|
作者
KLINGHOFER, V [1 ]
BAROW, JL [1 ]
STEIN, HH [1 ]
COHEN, J [1 ]
ROSENBERG, SH [1 ]
BAKER, WR [1 ]
VERBURG, KM [1 ]
POLAKOWSKI, JS [1 ]
KLEINERT, HD [1 ]
机构
[1] ABBOTT LABS, ABBOTT PK, IL 60064 USA
来源
FASEB JOURNAL | 1992年 / 6卷 / 05期
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:A1871 / A1871
页数:1
相关论文
共 50 条
  • [1] ABBOTT-72517 - A POTENT INHIBITOR OF RENIN WITH HYPOTENSIVE ACTIVITY IN THE DOG
    STEIN, HH
    ROSENBERG, SH
    BAKER, WR
    COHEN, J
    DAYTON, BD
    VERBURG, KM
    POLAKOWSKI, JS
    KLEINERT, HD
    FASEB JOURNAL, 1992, 6 (05): : A1870 - A1870
  • [2] DETECTION OF NANOGRAM LEVELS OF ORALLY ACTIVE RENIN INHIBITOR ABBOTT-72517 IN DOG PLASMA USING A RENIN INHIBITOR ACTIVITY ASSAY - COMPARISON TO HPLC RESULTS
    BARLOW, JL
    KLINGHOFER, V
    STEIN, HH
    ROSENBERG, SH
    BAKER, WR
    VERBURG, KM
    POLAKOWSKI, JS
    KLEINERT, HD
    FASEB JOURNAL, 1992, 6 (05): : A1870 - A1870
  • [3] RENIN INHIBITOR, ABBOTT-72517, DOES NOT INDUCE CHARACTERISTIC ANGIOTENSIN-CONVERTING ENZYME-INHIBITOR (ACEI) COUGH
    NELSON, DE
    MOYSE, DM
    ONEIL, JM
    BOGER, RS
    GLASSMAN, HN
    KLEINERT, HD
    CIRCULATION, 1993, 88 (04) : 361 - 361
  • [4] Zankiren (A-72517): Design of a peptide-derived, orally active renin inhibitor
    Rosenberg, SH
    Spina, KP
    Polakowski, J
    Kovar, P
    Stein, H
    Cohen, J
    Egan, DA
    Barlow, JL
    Klinghofer, V
    Hoffman, DJ
    Baker, WR
    Kleinert, HD
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 211 : 9 - BTEC
  • [5] CARDIOVASCULAR PROFILE OF THE ORALLY ACTIVE RENIN INHIBITOR A-72517 IN SODIUM-DEPLETED DOGS
    WESSALE, JL
    CALZADILLA, SV
    KOVAR, PJ
    ROSENBERG, SH
    BAKER, WR
    KLEINERT, HD
    FASEB JOURNAL, 1992, 6 (05): : A1871 - A1871
  • [6] AN ORALLY ACTIVE INHIBITOR OF RENIN
    PALS, DT
    THAISRIVONGS, S
    LAWSON, JA
    KATI, WM
    TURNER, SR
    DEGRAAF, GL
    HARRIS, DW
    JOHNSON, GA
    HYPERTENSION, 1986, 8 (12) : 1105 - 1112
  • [7] AN ORALLY-ACTIVE INHIBITOR OF RENIN
    PALS, DT
    THAISRIVONGS, S
    LAWSON, JA
    KATI, WM
    TURNER, SR
    DEGRAAF, GL
    HARRIS, DW
    JOHNSON, GA
    HYPERTENSION, 1986, 8 (09) : 833 - 833
  • [8] AN ORALLY ACTIVE INHIBITOR OF HUMAN RENIN
    KOKUBU, T
    HIWADA, K
    MURAKAMI, E
    MUNETA, S
    KITAMI, Y
    MORISAWA, Y
    KOIKE, H
    TAKAHAGI, H
    IIJIMA, Y
    NISHIMURA, K
    SALMON, PF
    HYPERTENSION, 1989, 14 (03) : 357 - 357
  • [9] Aliskiren: An orally active renin inhibitor
    Wal, Pranay
    Wal, Ankita
    Rai, Awani K.
    Dixit, Anuj
    JOURNAL OF PHARMACY AND BIOALLIED SCIENCES, 2011, 3 (02): : 189 - 193
  • [10] Pharmacokinetics of remikiren, a potent orally active inhibitor of human renin, in rat, dog and primates
    Coassolo, P
    Fischli, W
    Clozel, JP
    Chou, RC
    XENOBIOTICA, 1996, 26 (03) : 333 - 345