THE DOPAMINE UPTAKE INHIBITOR GBR 12909 - SELECTIVITY AND MOLECULAR MECHANISM OF ACTION

被引:356
作者
ANDERSEN, PH
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D O I
10.1016/0014-2999(89)90363-4
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:493 / 504
页数:12
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[2]   A COMPARISON BETWEEN DOPAMINE-STIMULATED ADENYLATE-CYCLASE AND H-3-SCH-23390 BINDING IN RAT STRIATUM [J].
ANDERSEN, PH ;
GRONVALD, FC ;
JANSEN, JA .
LIFE SCIENCES, 1985, 37 (21) :1971-1983
[3]  
ANDERSEN PH, 1986, ACTA PHARMACOL TOX, V59, P1315
[4]  
ANDERSENPH, 1987, 10TH IUPHAR SYDN
[5]   COEXISTENCE OF CARRIERS FOR DOPAMINE AND GABA UPTAKE ON A SAME NERVE-TERMINAL IN THE RAT-BRAIN [J].
BONANNO, G ;
RAITERI, M .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 91 (01) :237-243
[6]   HIGH-AFFINITY [H-3] GBR 12783 BINDING TO A SPECIFIC SITE ASSOCIATED WITH THE NEURONAL DOPAMINE UPTAKE COMPLEX IN THE CENTRAL-NERVOUS-SYSTEM [J].
BONNET, JJ ;
PROTAIS, P ;
CHAGRAOUI, A ;
COSTENTIN, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 126 (03) :211-222
[7]   GBR-12783, A POTENT AND SELECTIVE INHIBITOR OF DOPAMINE UPTAKE - BIOCHEMICAL-STUDIES INVIVO AND EXVIVO [J].
BONNET, JJ ;
COSTENTIN, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 121 (02) :199-209
[8]   INTERACTION OF PITRAZEPIN WITH THE GABA BENZODIAZEPINE RECEPTOR COMPLEX AND WITH GLYCINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 118 (1-2) :115-121
[9]  
CALLIGARO DO, 1987, J PHARMACOL EXP THER, V243, P61
[10]  
COOPER BR, 1980, J PHARMACOL EXP THER, V215, P127