Libraries of functionalized small-molecule fragments that can be screened in whole cells could take phenotypic drug discovery to the next level, providing new opportunities against undertargeted proteins.
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Vrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, NetherlandsVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Blaazer, Antoni R.
Orrling, Kristina M.
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Vrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, NetherlandsVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Orrling, Kristina M.
Shanmugham, Anitha
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IOTA Pharmaceut, Cambridge, EnglandVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Shanmugham, Anitha
Jansen, Chimed
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Vrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, NetherlandsVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Jansen, Chimed
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Maes, Louis
Edink, Ewald
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Vrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, NetherlandsVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Edink, Ewald
Sterk, Geert Jan
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Vrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, NetherlandsVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Sterk, Geert Jan
Siderius, Marco
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Vrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, NetherlandsVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Siderius, Marco
England, Paul
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IOTA Pharmaceut, Cambridge, EnglandVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
England, Paul
Bailey, David
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IOTA Pharmaceut, Cambridge, EnglandVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
Bailey, David
de Esch, Iwan J. P.
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Vrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, NetherlandsVrije Univ Amsterdam, AIMMS, Fac Sci, Div Med Chem, NL-1081 HV Amsterdam, Netherlands
机构:
SCAI, German Natl Res Ctr Informat Technol, GMD, D-53754 St Augustin, GermanySCAI, German Natl Res Ctr Informat Technol, GMD, D-53754 St Augustin, Germany
Lemmen, C
Lengauer, T
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SCAI, German Natl Res Ctr Informat Technol, GMD, D-53754 St Augustin, GermanySCAI, German Natl Res Ctr Informat Technol, GMD, D-53754 St Augustin, Germany
Lengauer, T
MOLECULAR MODELING AND PREDICTION OF BIOACTIVITY,
2000,
: 169
-
174
机构:Univ Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Morley, Andrew D.
Pugliese, Angelo
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Beatson Inst Canc Res, Glasgow G61 1BD, Lanark, ScotlandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Pugliese, Angelo
Birchall, Kristian
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Med Res Council Technol, London NW7 1AD, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Birchall, Kristian
Bower, Justin
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Beatson Inst Canc Res, Glasgow G61 1BD, Lanark, ScotlandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Bower, Justin
Brennan, Paul
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Struct Genom Consortium, Oxford 0X3 7DQ, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Brennan, Paul
Brown, Nathan
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Inst Canc Res, Div Canc Therapeut, Canc Res UK Canc Therapeut Unit, Sutton SM2 5NG, Surrey, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Brown, Nathan
Chapman, Tim
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Med Res Council Technol, London NW7 1AD, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Chapman, Tim
Drysdale, Martin
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Beatson Inst Canc Res, Glasgow G61 1BD, Lanark, ScotlandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Drysdale, Martin
Gilbert, Ian H.
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机构:Univ Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Gilbert, Ian H.
Hoelder, Swen
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Inst Canc Res, Div Canc Therapeut, Canc Res UK Canc Therapeut Unit, Sutton SM2 5NG, Surrey, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Hoelder, Swen
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Jordan, Allan
Ley, Steven V.
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Univ Cambridge, Dept Chem, Cambridge CB2 1EW, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Ley, Steven V.
Merritt, Andy
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Med Res Council Technol, London NW7 1AD, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Merritt, Andy
Miller, David
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UCL, London WC1E 6BT, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Miller, David
Swarbrick, Martin E.
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Canc Res Technol, Cambridge CB22 3AT, EnglandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland
Swarbrick, Martin E.
Wyatt, Paul G.
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Univ Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, ScotlandUniv Dundee, Coll Life Sci, Sir James Black Ctr, Dundee DD1 5EH, Scotland