68Ga-labeled cyclic RGD dimers with Gly3 and PEG4 linkers: promising agents for tumor integrin αvβ3 PET imaging

被引:0
|
作者
Zhaofei Liu
Gang Niu
Jiyun Shi
Shuanglong Liu
Fan Wang
Shuang Liu
Xiaoyuan Chen
机构
[1] Stanford University,Molecular Imaging Program at Stanford (MIPS), Department of Radiology, Biophysics & Bio
[2] Peking University,X
[3] Purdue University,Medical Isotopes Research Center
[4] Stanford University School of Medicine,School of Health Sciences
关键词
Integrin α; β; Ga; Bivalency; Angiogenesis molecular imaging targeting; PET tracer; Small animal PET;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:947 / 957
页数:10
相关论文
共 50 条
  • [1] 68Ga-labeled cyclic RGD dimers with Gly3 and PEG4 linkers: promising agents for tumor integrin αvβ3 PET imaging
    Liu, Zhaofei
    Niu, Gang
    Shi, Jiyun
    Liu, Shuanglong
    Wang, Fan
    Liu, Shuang
    Chen, Xiaoyuan
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2009, 36 (06) : 947 - 957
  • [2] Improving Tumor Uptake and Pharmacokinetics of 64Cu-Labeled Cyclic RGD Peptide Dimers with Gly3 and PEG4 Linkers
    Shi, Jiyun
    Kim, Young-Seung
    Zhai, Shizhen
    Liu, Zhaofei
    Chen, Xiaoyuan
    Liu, Shuang
    BIOCONJUGATE CHEMISTRY, 2009, 20 (04) : 750 - 759
  • [3] Preliminary biological evaluation of 68Ga-labeled cyclic RGD dimer as an integrin αvβ3-targeting radiotracer for tumor PET imaging
    Hui Ma
    Shaoyu Liu
    Zhanwen Zhang
    Ganghua Tang
    Gongjun Yuan
    Jing Zhao
    Shu Su
    Journal of Radioanalytical and Nuclear Chemistry, 2019, 321 : 857 - 865
  • [4] Preliminary biological evaluation of 68Ga-labeled cyclic RGD dimer as an integrin αvβ3-targeting radiotracer for tumor PET imaging
    Ma, Hui
    Liu, Shaoyu
    Zhang, Zhanwen
    Tang, Ganghua
    Yuan, Gongjun
    Zhao, Jing
    Su, Shu
    JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY, 2019, 321 (03) : 857 - 865
  • [5] In Vivo PET Imaging of the Cancer Integrin αvβ6 Using 68Ga-Labeled Cyclic RGD Nonapeptides
    Notni, Johannes
    Reich, Dominik
    Maltsev, Oleg V.
    Kapp, Tobias G.
    Steiger, Katja
    Hoffmann, Frauke
    Esposito, Irene
    Weichert, Wilko
    Kessler, Horst
    Wester, Hans-Juergen
    JOURNAL OF NUCLEAR MEDICINE, 2017, 58 (04) : 671 - 677
  • [6] 68Ga-labeled multimeric RGD peptides for microPET imaging of integrin αvβ3 expression
    Zi-Bo Li
    Kai Chen
    Xiaoyuan Chen
    European Journal of Nuclear Medicine and Molecular Imaging, 2008, 35 : 1100 - 1108
  • [7] 68Ga-labeled multimeric RGD peptides for microPET imaging of integrin αvβ3 expression
    Li, Zi-Bo
    Chen, Kai
    Chen, Xiaoyuan
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2008, 35 (06) : 1100 - 1108
  • [8] Improving tumor uptake and biodistribution characteristics of In-111-labeled cyclic RGD dimers with triglycine and PEG4 linkers
    Shi, Jin
    Kim, Young-Seung
    Zhai, Shizhen
    Jia, Bing
    Wang, Fan
    Liu, Shuang
    JOURNAL OF NUCLEAR MEDICINE, 2009, 50
  • [9] Improving Tumor-Targeting Capability and Pharmacokinetics of 99mTc-Labeled Cyclic RGD Dimers with PEG4 Linkers
    Wang, Lijun
    Shi, Jiyun
    Kim, Young-Seung
    Zhai, Shizhen
    Jia, Bing
    Zhao, Huiyun
    Liu, Zhaofei
    Wang, Fan
    Chen, Xiaoyuan
    Liu, Shuang
    MOLECULAR PHARMACEUTICS, 2009, 6 (01) : 231 - 245
  • [10] Evaluation of 68Ga-labeled RGD peptides for αvβ3 integrin detection in myocardial infarct
    Laitinen, Iina
    Pohle, Karolin
    Notni, Johannes
    Rudelius, Martina
    Weidl, Eliane
    Henriksen, Gjermund
    Wester, Hans
    Schwaiger, Markus
    JOURNAL OF NUCLEAR MEDICINE, 2012, 53