Synthesis and antifungal activity of sulfides, sulfoxides, and sulfones based on (1S)-(-)-β-pinene

被引：0
|
作者：
V. V. Gavrilov
V. A. Startseva
L. E. Nikitina
O. A. Lodochnikova
O. I. Gnezdilov
S. A. Lisovskaya
N. I. Glushko
E. N. Klimovitskii
机构：
[1] Kazan’ State University,A. M. Butlerov Chemical Institute
[2] Kazan’ State Medical University,A. E. Arbuzov Institute of Organic and Physical Chemistry, Kazan’ Scientific Center
[3] Russian Academy of Sciences,E. K. Zavoiskii Kazan’ Physicotechnical Institute, Kazan’ Scientific Center
[4] Russian Academy of Sciences,undefined
来源：
Pharmaceutical Chemistry Journal | 2010年 / 44卷
关键词：
Pinane sulfides; sulfoxides; and sulfones; antifungal activity;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Attachment of 2-mercaptoethanol and thioglycolic acid methyl ester to the double bond of (1S)-(-)-β-pinene yielded pinane sulfides with the cis configuration. Oxidation of sulfides with m-chloroperbenzoic acid yielded the corresponding sulfoxides and sulfones. The resulting compounds were screened for antimycotic activity and the dynamics of changes in antifungal properties in sulfides-sulfoxide-sulfone series were studied.
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页码：126 / 129
页数：3
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