NK3R antagonists: a novel approach for menopause symptoms

被引:0
|
作者
Simone Elder
Nanette Santoro
机构
[1] University of Colorado School of Medicine,Department of Obstetrics and Gynecology, Division of Reproductive Endocrinology
[2] Shady Grove Fertility,undefined
来源
关键词
D O I
暂无
中图分类号
学科分类号
摘要
Most women experience vasomotor symptoms during menopause, which considerably affect their quality of life. While vasomotor symptoms can be substantially reduced with menopausal hormone therapy, many women are unable or choose not to take hormone therapy. Now, studies have demonstrated that neurokinin 3 receptor antagonists have a level of effectiveness against vasomotor symptoms that is similar to that of hormone therapy.
引用
收藏
页码:617 / 618
页数:1
相关论文
共 50 条
  • [1] NK3R antagonists: a novel approach for menopause symptoms
    Elder, Simone
    Santoro, Nanette
    NATURE REVIEWS ENDOCRINOLOGY, 2023, 19 (11) : 617 - 618
  • [2] A Nonhormonal Selective NK3R Antagonist for Moderate to Severe Vasomotor Symptoms in Menopause
    不详
    CLINICAL NURSE SPECIALIST, 2023, 37 (06) : E5 - E5
  • [3] Fezolinetant: A novel NK3R antagonist for treating postmenopausal vasomotor symptoms
    Ali, Saqib
    Ilyas, Muhammad Affan
    JOURNAL OF THE PAKISTAN MEDICAL ASSOCIATION, 2024, 74 (08) : 1582 - 1582
  • [4] Neural Pathways of NK3R Inhibition in Vasomotor Symptoms
    Navarro, Victor M.
    MENOPAUSE-THE JOURNAL OF THE NORTH AMERICAN MENOPAUSE SOCIETY, 2023, 30 (12): : 1254 - 1254
  • [5] Update on NK3R antagonist fezolinetant
    Stute, P.
    GYNAKOLOGISCHE ENDOKRINOLOGIE, 2021, 19 (02): : 163 - 164
  • [6] Update NK3R-Antagonist FezolinetantUpdate on NK3R antagonist fezolinetant
    P. Stute
    Gynäkologische Endokrinologie, 2021, 19 : 163 - 164
  • [7] Development of Novel Neurokinin 3 Receptor (NK3R) Selective Agonists with Resistance to Proteolytic Degradation
    Misu, Ryosuke
    Oishi, Shinya
    Yamada, Ai
    Yamamura, Takashi
    Matsuda, Fuko
    Yamamoto, Koki
    Noguchi, Taro
    Ohno, Hiroaki
    Okamura, Hiroaki
    Ohkura, Satoshi
    Fujii, Nobutaka
    JOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (20) : 8646 - 8651
  • [8] Tacr3/NK3R: Beyond Their Roles in Reproduction
    Zhang, Wen-wen
    Wang, Yanqing
    Chu, Yu-Xia
    ACS CHEMICAL NEUROSCIENCE, 2020, 11 (19): : 2935 - 2943
  • [9] Heterologous desensitization and trafficking of neurokinin 1 and 3 receptors (NK1R, NK3R).
    Dery, O
    Lovett, M
    Grady, EF
    Bunnett, NW
    GASTROENTEROLOGY, 2000, 118 (04) : A304 - A304
  • [10] NK3R antagonist ameliorates metabolic status and reverses obesity in mice
    Shi, Y.
    Zhu, X.
    Liu, Y.
    HUMAN REPRODUCTION, 2019, 34 : 6 - 6