Synthesis of 3-acetyl-4-arylamino-2H-pyran-2-one derivatives

被引：0
|
作者：
Azuma, Y
Sato, A
Morone, M
机构：
[1] Tohoku College of Pharmacy, Aoba-ku, Sendai 981
来源：
YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN | 1997年 / 117卷 / 09期
关键词：
dehydroacetic acid; 2H-pyran-2-one; 3-acetyl-4-arylamino-6-methyl-2H-pyran-2-one; arylamination; beta-arylaminocarbonyl;
D O I：
10.1248/yakushi1947.117.9_618
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
A one-pot reaction of 4-chloro-3-(1-chlorovinyl)-6-methyl-2H-pyran-2-one with anilines in the presence of triethylamine gives 3-acetyl-4-arylamino-6-methyl-2H-pyran-2-one derivatives in good yields.
引用
收藏
页码：618 / 622
页数：5
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