BIOL 17-The MYST histone acetyltransferase TIP60: Mechanism, fluorescent reporters, and inhibitor discovery

被引:0
|
作者
Zheng, Yujun George [1 ]
机构
[1] Georgia State Univ, Dept Chem, Atlanta, GA 30302 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
17-BIOL
引用
收藏
页数:1
相关论文
共 50 条
  • [1] Rational design and validation of a Tip60 histone acetyltransferase inhibitor
    Gao, Chunxia
    Bourke, Emer
    Scobie, Martin
    Famme, Melina Arcos
    Koolmeister, Tobias
    Helleday, Thomas
    Eriksson, Leif A.
    Lowndes, Noel F.
    Brown, James A. L.
    SCIENTIFIC REPORTS, 2014, 4
  • [2] Rational design and validation of a Tip60 histone acetyltransferase inhibitor
    Chunxia Gao
    Emer Bourke
    Martin Scobie
    Melina Arcos Famme
    Tobias Koolmeister
    Thomas Helleday
    Leif A. Eriksson
    Noel F. Lowndes
    James A. L. Brown
    Scientific Reports, 4
  • [3] The MYST domain histone acetyltransferase TIP60 interacts with and is as a coactivator of the myeloid transcription factor C/EBPα.
    Bararia, Deepak
    Trivedi, Arun K.
    Zada, Abdul Peer
    Behre, Hermann M.
    Behre, Gerhard
    Bohlander, Stefan K.
    Dreyling, Martin H.
    BLOOD, 2006, 108 (11) : 163B - 163B
  • [4] Small molecule inhibitors of histone acetyltransferase Tip60
    Wu, Jiang
    Wang, Juxian
    Li, Minyong
    Yang, Yutao
    Wang, Binghe
    Zheng, Y. George
    BIOORGANIC CHEMISTRY, 2011, 39 (1-3) : 53 - 58
  • [5] Regulation of Histone Acetyltransferase TIP60 Function by Histone Deacetylase 3
    Yi, Jingjie
    Huang, Xiangyang
    Yang, Yuxia
    Zhu, Wei-Guo
    Gu, Wei
    Luo, Jianyuan
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2014, 289 (49) : 33878 - 33886
  • [6] A role for the Tip60 histone acetyltransferase in the acetylation and activation of ATM
    Sun, YL
    Jiang, XF
    Chen, SJ
    Fernandes, N
    Price, BD
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2005, 102 (37) : 13182 - 13187
  • [7] MYC recruits the TIP60 histone acetyltransferase complex to chromatin
    Frank, SR
    Parisi, T
    Taubert, S
    Fernandez, P
    Fuchs, M
    Chan, HM
    Livingston, DM
    Amati, B
    EMBO REPORTS, 2003, 4 (06) : 575 - 580
  • [8] The interaction of ETV6 (TEL) and TIP60 requires a functional histone acetyltransferase domain in TIP60
    Putnik, Jasmina
    Zhang, Chang-Dong
    Archangelo, Leticia Froehlich
    Tizazu, Belay
    Bartels, Sigrun
    Kickstein, Michael
    Greif, Philipp A.
    Bohlander, Stefan K.
    BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR BASIS OF DISEASE, 2007, 1772 (11-12): : 1211 - 1224
  • [9] Stratification of breast cancer patients using Tip60 staining paired with evaluation of a designed Tip60 specific histone acetyltransferase inhibitor for targeted treatment
    Shalaby, A.
    Emma, H.
    Bourke, E.
    Gao, C.
    Martin, S.
    Michael, K.
    Eriksson, L.
    Thomas, H.
    Brown, J.
    EUROPEAN JOURNAL OF CANCER, 2016, 61 : S130 - S130
  • [10] Putative involvement of the histone acetyltransferase Tip60 in ribosomal gene transcription
    Halkidou, K
    Logan, IR
    Cook, S
    Neal, DE
    Robson, CN
    NUCLEIC ACIDS RESEARCH, 2004, 32 (05) : 1654 - 1665