共 27 条
- [1] The mechanism of action of BT1718, a novel small-molecule drug conjugate for the treatment of solid tumors expressing MT1-MMPMOLECULAR CANCER THERAPEUTICS, 2018, 17 (01)Bennett, Gavin论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Cambridge, England Bicycle Therapeut Ltd, Cambridge, EnglandRigby, Mike论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Cambridge, England Bicycle Therapeut Ltd, Cambridge, EnglandLutz, Bob论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Cambridge, England Bicycle Therapeut Ltd, Cambridge, EnglandPark, Peter论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Cambridge, England Bicycle Therapeut Ltd, Cambridge, EnglandKeen, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Cambridge, England Bicycle Therapeut Ltd, Cambridge, England
- [2] Development of BT1718, a novel Bicycle Drug Conjugate for the treatment of lung cancerCANCER RESEARCH, 2017, 77Bennett, Gavin论文数: 0 引用数: 0 h-index: 0Lutz, Robert论文数: 0 引用数: 0 h-index: 0Park, Peter论文数: 0 引用数: 0 h-index: 0Harrison, Helen论文数: 0 引用数: 0 h-index: 0Lee, Kevin论文数: 0 引用数: 0 h-index: 0
- [3] BT1718, a novel bicyclic peptide-maytansinoid conjugate targeting MT1-MMP for the treatment of solid tumors: Design of bicyclic peptide and linker selectionCANCER RESEARCH, 2017, 77Harrison, Helen论文数: 0 引用数: 0 h-index: 0Bennett, Gavin论文数: 0 引用数: 0 h-index: 0Blakeley, Diane论文数: 0 引用数: 0 h-index: 0Brown, Amy论文数: 0 引用数: 0 h-index: 0Campbell, Spencer论文数: 0 引用数: 0 h-index: 0Chen, Liuhong论文数: 0 引用数: 0 h-index: 0Lutz, Robert J.论文数: 0 引用数: 0 h-index: 0Pavan, Silvia论文数: 0 引用数: 0 h-index: 0van Rietschoten, Katerine论文数: 0 引用数: 0 h-index: 0Teufel, Daniel论文数: 0 引用数: 0 h-index: 0Park, Peter U.论文数: 0 引用数: 0 h-index: 0Lee, Kevin论文数: 0 引用数: 0 h-index: 0
- [4] Preliminary pharmacokinetic assessment of BT1718: A phase I/IIa trial of BT1718 (a first in class Bicycle Toxin Conjugate) in patients with advanced solid tumoursEUROPEAN JOURNAL OF CANCER, 2018, 103 : E65 - E65Banerji, U.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton, Surrey, England Inst Canc Res, London, EnglandCook, N.论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Manchester, Lancs, England Christie NHS Fdn Trust, Christie Sch Oncol, Manchester, Lancs, England Inst Canc Res, London, EnglandEvans, T. R. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Glasgow, Glasgow, Lanark, Scotland Beatson West Scotland Canc Ctr, Canc Res Ctr, Glasgow, Lanark, Scotland Inst Canc Res, London, EnglandMoreno, I.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton, Surrey, England Inst Canc Res, London, EnglandPatricia, R.论文数: 0 引用数: 0 h-index: 0机构: Univ Glasgow, Glasgow, Lanark, Scotland Beatson West Scotland Canc Ctr, Canc Res Ctr, Glasgow, Lanark, Scotland Inst Canc Res, London, England论文数: 引用数: h-index:机构:Sabaratnam, N.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, England Inst Canc Res, London, EnglandPassi, R.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton, Surrey, England Inst Canc Res, Sutton, Surrey, England Inst Canc Res, London, EnglandGodfrey, L.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, Drug Dev, London, England Inst Canc Res, London, EnglandSawretse, L.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, Drug Dev, London, England Inst Canc Res, London, EnglandKatugampola, S.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, Drug Dev, London, England Inst Canc Res, London, EnglandHalbert, G.论文数: 0 引用数: 0 h-index: 0机构: Univ Strathclyde, Canc Res UK Formulat Unit, Glasgow, Lanark, Scotland Inst Canc Res, London, EnglandJeffrey, P.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Dev, Cambridge, England Inst Canc Res, London, EnglandRigby, M.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Dev, Cambridge, England Inst Canc Res, London, EnglandBennett, G.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Dev, Cambridge, England Inst Canc Res, London, EnglandKoehler, M.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Dev, Cambridge, England Inst Canc Res, London, EnglandLangford, G.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Dev, Cambridge, England Inst Canc Res, London, EnglandPittman, M.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, Drug Dev, London, England Inst Canc Res, London, EnglandSymeonides, S. N.论文数: 0 引用数: 0 h-index: 0机构: Univ Edinburgh, Edinburgh, Midlothian, Scotland Canc Res UK Ctr Drug Dev, London, England Canc Res UK Edinburgh Ctr, Edinburgh, Midlothian, Scotland Inst Canc Res, London, England
- [5] Pharmacokinetic (PK) assessment of BT1718: A phase I/II a study of BT1718, a first in class bicycle toxin conjugate (BTC), in patients (pts) with advanced solid tumoursANNALS OF ONCOLOGY, 2019, 30 : 174 - 174Cook, N.论文数: 0 引用数: 0 h-index: 0机构: Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandBanerji, U.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Inst Canc Res, Drug Dev Unit, Sutton, Surrey, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandEvans, J.论文数: 0 引用数: 0 h-index: 0机构: Beatson West Scotland Canc Ctr, Med Oncol, Glasgow, Lanark, Scotland Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandBiondo, A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Inst Canc Res, Drug Dev Unit, Sutton, Surrey, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandGermetaki, T.论文数: 0 引用数: 0 h-index: 0机构: Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandRandhawa, M.论文数: 0 引用数: 0 h-index: 0机构: Beatson West Scotland Canc Ctr, Med Oncol, Glasgow, Lanark, Scotland Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandGodfrey, L.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK, Ctr Drug Dev, London, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandLeslie, S.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK, Ctr Drug Dev, London, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandJeffrey, P.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Preclin Dev, Cambridge, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandRigby, M.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Preclin Dev, Cambridge, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandBennett, G.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Preclin Dev, Cambridge, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandBlakemore, S.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Translat Sci, Lexington, AL USA Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandKoehler, M.论文数: 0 引用数: 0 h-index: 0机构: REPARETherapeutics, Oncol, Cambridge, MA USA Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandNiewiarowski, A.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK, Ctr Drug Dev, London, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandPittman, M.论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK, Ctr Drug Dev, London, England Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, EnglandSymeonides, S. N.论文数: 0 引用数: 0 h-index: 0机构: Western Gen Hosp, Edinburgh Canc Ctr, Edinburgh, Midlothian, Scotland Christie NHS Fdn Trust, Dept Med Oncol, Manchester, Lancs, England
- [6] A Cancer Research UK phase I/IIa trial of BT1718 (a first in class Bicycle Drug Conjugate) given intravenously in patients with advanced solid tumours.JOURNAL OF CLINICAL ONCOLOGY, 2018, 36 (15)Banerji, Udai论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandCook, Natalie论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandEvans, T. R. Jeffry论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandCandilejo, Irene Moreno论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandRoxburgh, Patricia论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandKelly, Claire L. S.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandSabaratnam, Narmatha论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandPassi, Rashmi论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandLeslie, Sawretse论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandKatugampola, Sidath论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandGodfrey, Lisa论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandTremayne, Neil论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandBennett, Gavin论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandKoehler, Maria论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandLangford, Gillian论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandSymeonides, Stefan N.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, EnglandPittman, Marc论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England
- [7] A Cancer Research UK phase I/IIa trial of BT1718 (a first in class Bicycle Toxin Conjugate) given intravenously in patients with advanced solid tumoursBRITISH JOURNAL OF CANCER, 2018, 119 (11) : 42 - 42Banerji, Udai论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res Royal Marsden NHS Fdn Trust, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, England论文数: 引用数: h-index:机构:Evans, T. R. Jeffry论文数: 0 引用数: 0 h-index: 0机构: Univ Glasgow, Glasgow, Lanark, Scotland Beatson West Scotland Canc Ctr, Glasgow, Lanark, Scotland Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandCandilejo, Irene Moreno论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res Royal Marsden NHS Fdn Trust, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, England论文数: 引用数: h-index:机构:Kelly, Claire论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester Christie NHS Fdn Trust, Manchester, Lancs, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandSabaratnam, Narmatha论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res Royal Marsden NHS Fdn Trust, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandPassi, Rashmi论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res Royal Marsden NHS Fdn Trust, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandLeslie, Sawretse论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandKatugampola, Sidath论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandGodfrey, Lisa论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandTremayne, Neil论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandHalbert, Gavin论文数: 0 引用数: 0 h-index: 0机构: Univ Strathclyde, Canc Res UK Formulat Unit, Glasgow, Lanark, Scotland Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandBennett, Gavin论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandKoehler, Maria论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandLangford, Gillian论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandPittman, Marc论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, London, England Inst Canc Res Royal Marsden NHS Fdn Trust, London, EnglandSymeonides, Stefan论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Ctr Drug Dev, London, England Univ Edinburgh, Edinburgh, Midlothian, Scotland Inst Canc Res Royal Marsden NHS Fdn Trust, London, England
- [8] MT1-MMP Immunohistochemistry (IHC) analysis of tumor microarrays (TMAs) using a novel scoring system guides patient selection for BT1718 expansion cohortsMOLECULAR CANCER THERAPEUTICS, 2019, 18 (12)Gelb, Tara论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USABacon, Chris论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Northern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Bicycle Therapeut, Lexington, MA USASloan, Philip论文数: 0 引用数: 0 h-index: 0机构: Royal Victoria Infirm, Newcastle Mol Pathol Node, Newcastle Upon Tyne, Tyne & Wear, England Bicycle Therapeut, Lexington, MA USARigby, Mike论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Cambridge, England Bicycle Therapeut, Lexington, MA USAGuerrera, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USAKelly, Fiona论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK, Ctr Drug Dev, London, England Bicycle Therapeut, Lexington, MA USASymeonides, Stefan论文数: 0 引用数: 0 h-index: 0机构: Canc Res UK Edinburgh Ctr, Edinburgh, Midlothian, Scotland Bicycle Therapeut, Lexington, MA USABlakemore, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut, Lexington, MA USA Bicycle Therapeut, Lexington, MA USA
- [9] Design and characterization of a high affinity and selective bicyclic peptide binder to MT1-MMP for development of a treatment for solid tumoursEUROPEAN JOURNAL OF CANCER, 2016, 69 : S69 - S70Harrison, H.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Therapeut, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandChen, L.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Discovery, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandTeufel, D.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Therapeut, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandVan Rietschoten, K.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Discovery, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandCampbell, S.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Therapeut, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandBrown, A.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Therapeut, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandBlakeley, D.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Discovery, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandBennett, G.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Therapeut, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandLangford, G.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Therapeut, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, EnglandBonny, C.论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Ltd, Discovery, Cambridge, England Bicycle Therapeut Ltd, Therapeut, Cambridge, England
- [10] BT8009; A Nectin-4 Targeting Bicycle Toxin Conjugate for Treatment of Solid TumorsMOLECULAR CANCER THERAPEUTICS, 2022, 21 (12) : 1747 - 1756Rigby, Michael论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Blocks A&B,Portway Bldg,Granta Pk, Cambridge CB21 6GP, England Bicycle TX Ltd, Cambridge, EnglandBennett, Gavin论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandChen, Liuhong论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandMudd, Gemma E.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandHarrison, Helen论文数: 0 引用数: 0 h-index: 0机构: Amphista Therapeut, Cori Bldg, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandBeswick, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandVan Rietschoten, Katerine论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandWatcham, Sophie M.论文数: 0 引用数: 0 h-index: 0机构: Kymab Ltd, Bennet Bldg,Babraham Res Campus, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandScott, Heather S.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandBrown, Amy N.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandPark, Peter U.论文数: 0 引用数: 0 h-index: 0机构: Orum Therapeut, Cambridge, MA USA Bicycle TX Ltd, Cambridge, EnglandCampbell, Carly论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandHaines, Eric论文数: 0 引用数: 0 h-index: 0机构: Ikena Oncol, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandLahdenranta, Johanna论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandSkynner, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandJeffrey, Phil论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, EnglandKeen, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Bicycle Therapeut Inc, Boston, MA USA Bicycle TX Ltd, Cambridge, EnglandLee, Kevin论文数: 0 引用数: 0 h-index: 0机构: Bicycle TX Ltd, Cambridge, England Bicycle TX Ltd, Cambridge, England