Solid phase synthesis of 1,4-disubstituted 1,2,3-triazole from polystyrene-supported selenium resin

被引：0
|
作者：
Xu, Wei Ming
Wu, Lu Ling
Huang, Xian
机构：
[1] Zhejiang Univ, Dept Chem, Hangzhou 310028, Peoples R China
[2] Zhejiang Univ, Ctr Anal & Measurement, Hangzhou 310028, Peoples R China
来源：
CHINESE CHEMICAL LETTERS | 2006年 / 17卷 / 05期
关键词：
solid-phase synthesis; 1,3-dipolar cycloaddition; alpha-alkylation reaction; 1,2,3-triazole;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
We report here a solid-phase synthesis of 1, 4-disubstituted 1, 2, 3-triazole using polystyrene-supported selenium resin. The resin used here not only works as a simple linker, but also assists the crucial alpha-alkylation reaction and selenoxide syn-elimination, which ensures the purity of the products.
引用
收藏
页码：603 / 605
页数：3
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