首页
学术期刊
论文检测
AIGC检测
热点
更多
数据
Introduction: Human Metabolites in Safety Testing (MIST) Issue
被引:32
|
作者
:
Guengerich, F. Peter
论文数:
0
引用数:
0
h-index:
0
Guengerich, F. Peter
机构
:
来源
:
CHEMICAL RESEARCH IN TOXICOLOGY
|
2009年
/ 22卷
/ 02期
关键词
:
D O I
:
10.1021/tx900003k
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:237 / 238
页数:2
相关论文
共 50 条
[1]
Metabolites in Safety Testing: "MIST" for the Clinical Pharmacologist
Frederick, C. B.
论文数:
0
引用数:
0
h-index:
0
机构:
Merck Res Labs, Dept Safety Assessment, West Point, PA USA
Merck Res Labs, Dept Safety Assessment, West Point, PA USA
Frederick, C. B.
Obach, R. S.
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Global Res & Dev, Dept Pharmacokinet Pharmacodynam & Drug Metab, Groton, CT USA
Merck Res Labs, Dept Safety Assessment, West Point, PA USA
Obach, R. S.
CLINICAL PHARMACOLOGY & THERAPEUTICS,
2010,
87
(03)
: 345
-
350
[2]
LEVERAGING ADME DATA IN METABOLITES IN SAFETY TESTING (MIST)
Smith, Dennis Allen
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Global R&D, Dept PDM IPC 326, Sandwich, Kent, England
Pfizer Global R&D, Dept PDM IPC 326, Sandwich, Kent, England
Smith, Dennis Allen
Obach, R. Scott
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Global Res & Dev, Groton, CT USA
Pfizer Global R&D, Dept PDM IPC 326, Sandwich, Kent, England
Obach, R. Scott
DRUG METABOLISM REVIEWS,
2007,
39
: 31
-
31
[3]
Meeting Report: Metabolites in Safety Testing (MIST) Symposium—Safety Assessment of Human Metabolites: What’s REALLY Necessary to Ascertain Exposure Coverage in Safety Tests?
Hongying Gao
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc.,Pharmacokinetics, Dynamics and Metabolism
Hongying Gao
Abigail Jacobs
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc.,Pharmacokinetics, Dynamics and Metabolism
Abigail Jacobs
Ronald E. White
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc.,Pharmacokinetics, Dynamics and Metabolism
Ronald E. White
Brian P. Booth
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc.,Pharmacokinetics, Dynamics and Metabolism
Brian P. Booth
R. Scott Obach
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc.,Pharmacokinetics, Dynamics and Metabolism
R. Scott Obach
The AAPS Journal,
2013,
15
: 970
-
973
[4]
Meeting Report: Metabolites in Safety Testing (MIST) Symposium-Safety Assessment of Human Metabolites: What's REALLY Necessary to Ascertain Exposure Coverage in Safety Tests?
Gao, Hongying
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Pharmacokinet Dynam & Metab, Groton, CT 06340 USA
Pfizer Inc, Pharmacokinet Dynam & Metab, Groton, CT 06340 USA
Gao, Hongying
Jacobs, Abigail
论文数:
0
引用数:
0
h-index:
0
机构:
US FDA, Off New Drugs, Ctr Drug Evaluat & Res, Silver Spring, MD USA
Pfizer Inc, Pharmacokinet Dynam & Metab, Groton, CT 06340 USA
Jacobs, Abigail
White, Ronald E.
论文数:
0
引用数:
0
h-index:
0
机构:
XenoBiot Labs Inc, DMPK Sci & Technol, Plainsboro, NJ USA
Pfizer Inc, Pharmacokinet Dynam & Metab, Groton, CT 06340 USA
White, Ronald E.
Booth, Brian P.
论文数:
0
引用数:
0
h-index:
0
机构:
US FDA, OTS OCP DCP V, Ctr Drug Evaluat & Res, Silver Spring, MD USA
Pfizer Inc, Pharmacokinet Dynam & Metab, Groton, CT 06340 USA
Booth, Brian P.
Obach, R. Scott
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Pharmacokinet Dynam & Metab, Groton, CT 06340 USA
Pfizer Inc, Pharmacokinet Dynam & Metab, Groton, CT 06340 USA
Obach, R. Scott
AAPS JOURNAL,
2013,
15
(04):
: 970
-
973
[5]
Metabolites in Safety Testing (MIST): Considerations of Mechanisms of Toxicity with Dose, Abundance, and Duration of Treatment
Smith, Dennis A.
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich, Kent, England
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich, Kent, England
Smith, Dennis A.
Obach, R. Scott
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Dynam & Metab, Groton, CT 06340 USA
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich, Kent, England
Obach, R. Scott
CHEMICAL RESEARCH IN TOXICOLOGY,
2009,
22
(02)
: 267
-
279
[6]
Seeing through the mist:: Abundance versus percentage.: Commentary on Metabolites in safety testing
Smith, DA
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Smith, DA
Obach, RS
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Obach, RS
DRUG METABOLISM AND DISPOSITION,
2005,
33
(10)
: 1409
-
1417
[7]
Why I love metabolites in safety testing (MIST): a light-hearted historical perspective
Tonelli, Alfred
论文数:
0
引用数:
0
h-index:
0
机构:
Johnson & Johnson Pharmaceut Res & Dev, Global Preclin Dev, Raritan, NJ USA
Johnson & Johnson Pharmaceut Res & Dev, External Res & Early Dev, Raritan, NJ USA
Johnson & Johnson Pharmaceut Res & Dev, Global Preclin Dev, Raritan, NJ USA
Tonelli, Alfred
BIOANALYSIS,
2009,
1
(04)
: 683
-
685
[8]
Clearing the MIST (metabolites in safety testing) of time: The impact of duration of administration on drug metabolite toxicity
Smith, Dennis A.
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Smith, Dennis A.
Obach, R. Scott
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Obach, R. Scott
Williams, Dominic P.
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3BX, Merseyside, England
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Williams, Dominic P.
Park, B. Kevin
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Liverpool, Dept Pharmacol & Therapeut, Liverpool L69 3BX, Merseyside, England
Pfizer Inc, Pharmacokinet Dynam & Metab, Sandwich CT13 9NJ, Kent, England
Park, B. Kevin
CHEMICO-BIOLOGICAL INTERACTIONS,
2009,
179
(01)
: 60
-
67
[9]
A Decade in the MIST: Learnings from Investigations of Drug Metabolites in Drug Development under the "Metabolites in Safety Testing" Regulatory Guidance
Schadt, Simone
论文数:
0
引用数:
0
h-index:
0
机构:
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Schadt, Simone
Bister, Bojan
论文数:
0
引用数:
0
h-index:
0
机构:
Boehringer Ingelheim Pharma GmbH & Co KG, Biberach, Germany
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Bister, Bojan
Chowdhury, Swapan K.
论文数:
0
引用数:
0
h-index:
0
机构:
Takeda Pharmaceut Int Co, Drug Metab & Pharmacokinet Dept, Cambridge, MA USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Chowdhury, Swapan K.
Funk, Christoph
论文数:
0
引用数:
0
h-index:
0
机构:
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Funk, Christoph
Hop, Cornelis E. C. A.
论文数:
0
引用数:
0
h-index:
0
机构:
Genentech Inc, Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Hop, Cornelis E. C. A.
Humphreys, W. Griffith
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol Myers Squibb Pharmaceut Co, Princeton, NJ USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Humphreys, W. Griffith
Igarashi, Fumihiko
论文数:
0
引用数:
0
h-index:
0
机构:
Chugai Pharmaceut Co Ltd, Res Div, Gotemba, Japan
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Igarashi, Fumihiko
James, Alexander D.
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst Biomed Res, PK Sci ADME, Basel, Switzerland
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
James, Alexander D.
Kagan, Mark
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst Biomed Res, PK Sci ADME, One Hlth Plaza, E Hanover, NJ USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Kagan, Mark
Khojasteh, S. Cyrus
论文数:
0
引用数:
0
h-index:
0
机构:
Genentech Inc, Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Khojasteh, S. Cyrus
Nedderman, Angus N. R.
论文数:
0
引用数:
0
h-index:
0
机构:
Unilabs York Bioanalyt Solut, Discovery Pk House,Discovery Pk, Sandwich, Kent, England
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Nedderman, Angus N. R.
Prakash, Chandra
论文数:
0
引用数:
0
h-index:
0
机构:
Agios, Drug Metab Pharmacokinet & Clin Pharmacol, Cambridge, MA USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Prakash, Chandra
Runge, Frank
论文数:
0
引用数:
0
h-index:
0
机构:
Boehringer Ingelheim Pharma GmbH & Co KG, Biberach, Germany
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Runge, Frank
Scheible, Holger
论文数:
0
引用数:
0
h-index:
0
机构:
NCE Drug Disposit, Merck Biopharma Quantitat Pharmacol & Drug Dispos, Darmstadt, Germany
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Scheible, Holger
Spracklin, Douglas K.
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer, Pharmacokinet Dynam & Metab, Groton, CT USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Spracklin, Douglas K.
Swart, Piet
论文数:
0
引用数:
0
h-index:
0
机构:
NCE Drug Disposit, Merck Biopharma Quantitat Pharmacol & Drug Dispos, Darmstadt, Germany
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Swart, Piet
Tse, Susanna
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer, Pharmacokinet Dynam & Metab, Groton, CT USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Tse, Susanna
Yuan, Josh
论文数:
0
引用数:
0
h-index:
0
机构:
Takeda Pharmaceut Int Co, Drug Metab & Pharmacokinet Dept, Cambridge, MA USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Yuan, Josh
Obach, R. Scott
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer, Pharmacokinet Dynam & Metab, Groton, CT USA
F Hoffmann La Roche Ltd, Roche Innovat Ctr Basel, Roche Pharma Res & Early Dev, Pharmaceut Sci, Grenzacher Str 124, CH-4070 Basel, Switzerland
Obach, R. Scott
DRUG METABOLISM AND DISPOSITION,
2018,
46
(06)
: 865
-
878
[10]
Addressing MIST (Metabolites in Safety Testing): Bioanalytical Approaches to Address Metabolite Exposures in Humans and Animals
Gao, Hongying
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Groton, CT 06340 USA
Pfizer Inc, Groton, CT 06340 USA
Gao, Hongying
Obach, R. Scott
论文数:
0
引用数:
0
h-index:
0
机构:
Pfizer Inc, Groton, CT 06340 USA
Pfizer Inc, Groton, CT 06340 USA
Obach, R. Scott
CURRENT DRUG METABOLISM,
2011,
12
(06)
: 578
-
586
←
1
2
3
4
5
→