Synthesis of chalcones, pyrazolines, amino pyrimidines and pyrimidinethiones as antibacterial agents

被引：0
|
作者：
Solankee, A [1 ]
Patel, J [1 ]
机构：
[1] BKM Sci Coll, Dept Chem, Valsad 396001, India
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2004年 / 43卷 / 07期
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中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
2-Phenylamino-4-(3'-fluorophenylamino)-6-(4'-acetylphenylamino)-s-triazine 5 on treatment with aromatic aldehydes yields chalcones 6a-f, which on cyclization with hydrazine hydrate, guanidine nitrate and thiourea give the corresponding pyrazolines 7a-f, amino pyrimidines 8a-f and pyrimidinethiones 9a-f, respectively. The synthesized compounds are screened for their antibacterial activity.
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页码：1580 / 1584
页数：5
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