Inhibition of the Staphylococcus aureus sortase transpeptidase SRTA by phosphinic peptidomimetics.

被引:0
|
作者
McCafferty, DG
Kruger, RG
Barkallah, S
Frankel, BA
机构
[1] Univ Penn, Sch Med, Dept Biochem & Biophys, Philadelphia, PA 19104 USA
[2] Univ Penn, Sch Med, Johnson Res Fdn, Philadelphia, PA 19104 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
198-BIOL
引用
收藏
页码:U203 / U204
页数:2
相关论文
共 50 条
  • [1] Inhibition of the Staphylococcus aureus sortase transpeptidase SrtA by phosphinic peptidomimetics
    Kruger, RG
    Barkallah, S
    Frankel, BA
    McCafferty, DG
    BIOORGANIC & MEDICINAL CHEMISTRY, 2004, 12 (13) : 3723 - 3729
  • [2] Irreversible inhibition of the Staphylococcus aureus transpeptidase sortase (SrtA) by vinyl sulfones
    Frankel, BA
    Otvos, B
    He, S
    Kruger, R
    McCafferty, DG
    BIOCHEMISTRY, 2003, 42 (28) : 8630 - 8630
  • [3] Analysis of the substrate specificity of the Staphylococcus aureus sortase transpeptidase SrtA
    Kruger, RG
    Otvos, B
    Frankel, BA
    Bentley, M
    Dostal, P
    McCafferty, DG
    BIOCHEMISTRY, 2004, 43 (06) : 1541 - 1551
  • [4] Evidence for a reverse protonation catalytic mechanism for the Staphylococcus aureus sortase transpeptidase SrtA
    Frankel, BA
    McCafferty, DG
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U607 - U607
  • [5] Kinetic mechanism of Staphylococcus aureus sortase SrtA
    Huang, XY
    Aulabaugh, A
    Ding, WD
    Kapoor, B
    Alksne, L
    Tabei, K
    Ellestad, G
    BIOCHEMISTRY, 2003, 42 (38) : 11307 - 11315
  • [6] Analysis of activity, substrate specificity, and kinetic mechanism of the Staphylococcus aureus sortase transpeptidase SrtA.
    Kruger, RG
    Otvos, B
    Dostal, PJ
    Frankel, BA
    Robinson, D
    Kelleher, NL
    McCafferty, DG
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2003, 226 : U153 - U153
  • [7] Analysis of activity, substrate specificity, and kinetic mechanism of the Staphylococcus aureus sortase transpeptidase SrtA.
    Kruger, RG
    Otvos, B
    Dostal, PJ
    Frankel, BA
    Robinson, D
    Kelleher, NL
    McCafferty, DG
    BIOCHEMISTRY, 2003, 42 (28) : 8599 - 8599
  • [8] Irreversible inhibition of the Staphylococcus aureus transpeptioase sortase (SRTA) by vinyl sulfones.
    Frankel, BA
    Otvos, B
    He, S
    Kruger, R
    McCafferty, DG
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2003, 226 : U176 - U176
  • [9] Staphylococcus aureus sortase transpeptidase SrtA:: Insight into the kinetic mechanism and evidence for a reverse protonation catalytic mechanism
    Frankel, BA
    Kruger, RG
    Robinson, DE
    Kelleher, NL
    McCafferty, DG
    BIOCHEMISTRY, 2005, 44 (33) : 11188 - 11200
  • [10] Development of a high-performance liquid chromatography assay and revision of kinetic parameters for the Staphylococcus aureus sortase transpeptidase SrtA
    Kruger, RG
    Dostal, P
    McCafferty, DG
    ANALYTICAL BIOCHEMISTRY, 2004, 326 (01) : 42 - 48