共 50 条
- [1] DESIGN AND SYNTHESIS OF POTENT, ORALLY BIOAVAILABLE HIV-1 PROTEASE INHIBITORSABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1994, 208 : 17 - MEDIKALDOR, SW论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121KALISH, V论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121DRESSMAN, BA论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121FRITZ, JE论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121HAMMOND, M论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121CROWELL, TA论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121TATLOCK, J论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121REICH, S论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121DAVIES, J论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121APPELT, K论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121SHETTY, B论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121SU, KS论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121CAMPANALE, KM论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121BURGESS, JA论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121LUBBENHUSEN, PP论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121BAXTER, AJ论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121MUESING, MA论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121HATCH, SD论文数: 0 引用数: 0 h-index: 0机构: AGOURON PHARMACEUT INC,SAN DIEGO,CA 92121
- [2] SPECIFIC HIV-1 INHIBITORS TARGETED AT THE HIV-1 RTJOURNAL OF ACQUIRED IMMUNE DEFICIENCY SYNDROMES AND HUMAN RETROVIROLOGY, 1993, 6 (06): : 673 - 673DECLERCQ, E论文数: 0 引用数: 0 h-index: 0机构: CATHOLIC UNIV LEUVEN,REGA INST MED RES,B-3000 LOUVAIN,BELGIUM CATHOLIC UNIV LEUVEN,REGA INST MED RES,B-3000 LOUVAIN,BELGIUM
- [3] Design and synthesis of novel and potent allosteric HIV-1 integrase inhibitors with a spirocyclic moietyBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 110Adachi, Kaoru论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanManabe, Tomoyuki论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Innovat Implementat Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanYamasaki, Takayuki论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Dept Res Planning, Preclin, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanSuma, Akira论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Innovat Implementat Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanOrita, Takuya论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanFuruzono, Tomoko论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanAdachi, Tsuyoshi论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanOhata, Yoshitsugu论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Biol Pharmacol Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanAkiyama, Yoshiyuki论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, DMPK Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, JapanMiyazaki, Susumu论文数: 0 引用数: 0 h-index: 0机构: Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan Japan Tobacco Inc, Cent Pharmaceut Res Inst, Chem Res Labs, 1-1,Murasaki Cho, Takatsuki, Osaka 5691125, Japan
- [4] Design and synthesis of bicyclic pyrimidinones as potent and orally bioavailable HIV-1 integrase inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2008, 51 (04) : 861 - 874Muraglia, Ester论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyKinzel, Olaf论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyGardelli, Cristina论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyCrescenzi, Benedetta论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyDonghi, Monica论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyFerrara, Marco论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyNizi, Emanuela论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyOrvieto, Federica论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyPescatore, Giovanna论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyLaufer, Ralph论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyGonzalez-Paz, Odalys论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyDi Marco, Annalise论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyFiore, Fabrizio论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyMonteagudo, Edith论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyFonsi, Massimiliano论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalyFelock, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA USA IRBM, Merck Res Labs, I-00040 Pomezia, ItalyRowley, Michael论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, ItalySumma, Vincenzo论文数: 0 引用数: 0 h-index: 0机构: IRBM, Merck Res Labs, I-00040 Pomezia, Italy IRBM, Merck Res Labs, I-00040 Pomezia, Italy
- [5] Synthesis of 1-(alkyl)-5-dimethylamino-6-phenethyluracils as potent nonnucleoside HIV-1 RT inhibitorsSYNTHETIC COMMUNICATIONS, 2007, 37 (14) : 2421 - 2431Wang, Xiaowei论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100083, Peoples R China Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100083, Peoples R ChinaChen, Yanli论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100083, Peoples R ChinaGuo, Ying论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100083, Peoples R ChinaLi, Amin论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100083, Peoples R ChinaMa, Xiaoyan论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100083, Peoples R ChinaLiu, Junyi论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100083, Peoples R China
- [6] 3 NEW POTENT HIV-1 INHIBITORS FROM MYXOBACTERIAANTIVIRAL CHEMISTRY & CHEMOTHERAPY, 1992, 3 (04): : 189 - 193JURKIEWICZ, E论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANYJANSEN, R论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANYKUNZE, B论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANYTROWITZSCHKIENAST, W论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANYFORCHE, E论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANYREICHENBACH, H论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANYHOFLE, G论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANYHUNSMANN, G论文数: 0 引用数: 0 h-index: 0机构: GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY GESELL BIOTECHNOL FORSCH GMBH,W-3300 BRAUNSCHWEIG,GERMANY
- [7] Design, synthesis and SAR study of bridged tricyclic pyrimidinone carboxamides as HIV-1 integrase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2020, 28 (13)Patel, Manoj论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USA ViiV Healthcare, 36 East Ind Pkwy, Branford, CT 06405 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USANaidu, B. Narasimhulu论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USA ViiV Healthcare, 36 East Ind Pkwy, Branford, CT 06405 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USADicker, Ira论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Virol, 5 Res Pkwy, Wallingford, CT 06492 USA ViiV Healthcare, 36 East Ind Pkwy, Branford, CT 06405 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAHigley, Helen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Virol, 5 Res Pkwy, Wallingford, CT 06492 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USALin, Zeyu论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Virol, 5 Res Pkwy, Wallingford, CT 06492 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USATerry, Brian论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Virol, 5 Res Pkwy, Wallingford, CT 06492 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAProtack, Tricia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Virol, 5 Res Pkwy, Wallingford, CT 06492 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAKrystal, Mark论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Virol, 5 Res Pkwy, Wallingford, CT 06492 USA ViiV Healthcare, 36 East Ind Pkwy, Branford, CT 06405 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAJenkins, Susan论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USA ViiV Healthcare, 36 East Ind Pkwy, Branford, CT 06405 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAParker, Dawn论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USA ViiV Healthcare, 36 East Ind Pkwy, Branford, CT 06405 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAPanja, Chiradeep论文数: 0 引用数: 0 h-index: 0机构: Biocon Bristol Myers Squibb Res Ctr, Plot 2&3,Bommasandra Ind Estate Phase 4, Bengaluru 560099, Karnataka, India Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USARampulla, Richard论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Dept Discovery Chem Synth, POB 4000, Princeton, NJ 08543 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAMathur, Arvind论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Dept Discovery Chem Synth, POB 4000, Princeton, NJ 08543 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAMeanwell, Nicholas A.论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USAWalker, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USA Assembly Biosci Inc, 331 Oyster Point Blvd, San Francisco, CA 94080 USA Dept Discovery Chem & Mol Technol, 5 Res Pkwy, Wallingford, CT 06492 USA
- [8] Synthesis of a new class of HIV-1 inhibitorsNUCLEOSIDES & NUCLEOTIDES, 1999, 18 (02): : 263 - 275Farese-Di Giorgio, A论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, FrancePairot, S论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, FrancePatino, N论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, FranceCondom, R论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, France Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, FranceDi Giorgio, C论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, FranceAumelas, A论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, FranceAubertin, AM论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, FranceGuedj, R论文数: 0 引用数: 0 h-index: 0机构: Univ Nice, Chim Bioorgan Lab, CNRS ESA 6001, F-06108 Nice 2, France
- [9] Design and Synthesis of Piperazine Sulfonamide Cores Leading to Highly Potent HIV-1 Protease InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2017, 8 (12): : 1292 - 1297Bungard, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAWilliams, Peter D.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USASchulz, Jurgen论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAWiscount, Catherine M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAHolloway, M. Katharine论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USALoughran, H. Marie论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAManikowski, Jesse J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USASu, Hua-Poo论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USABennett, David J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAChang, Lehua论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAChu, Xin-Jie论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USACrespo, Alejandro论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USADwyer, Michael P.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAKeertikar, Kartik论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAMorriello, Gregori J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAStamford, Andrew W.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAWaddell, Sherman T.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAZhong, Bin论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAHu, Bin论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAJo, Tao论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USADiamond, Tracy L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USABahnck-Teets, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USACarroll, Steven S.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAFay, John F.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAMin, Xu论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAMorris, William论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 126 East Lincoln Ave, Rahway, NJ 07065 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USABallard, Jeanine E.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAMiller, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USAMcCauley, John A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA Merck & Co Inc, 770 Sumneytown Pike,POB 4, West Point, PA 19486 USA
- [10] Design, synthesis and SAR of thienopyridines as potent CHK1 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (24) : 7216 - 7221Zhao, Lianyun论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem, Cambridge, MA 02141 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USAZhang, Yingxin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem, Cambridge, MA 02141 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USADai, Chaoyang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem, Cambridge, MA 02141 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USAGuzi, Timothy论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem, Cambridge, MA 02141 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USAWiswell, Derek论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Palo Alto, CA 94304 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USASeghezzi, Wolfgang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Palo Alto, CA 94304 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USAParry, David论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Palo Alto, CA 94304 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USAFischmann, Thierry论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Design Dept, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USASiddiqui, M. Arshad论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem, Cambridge, MA 02141 USA Merck Res Labs, Dept Chem, Cambridge, MA 02141 USA