Synthesis of 8-[10B]-dihydroxyboryl-harmine, a potential agent for boron neutron capture therapy.

被引：0

作者：

Sintas, JA ^{[1
]}

Macareno, NJ ^{[1
]}

Vitale, AA ^{[1
]}

机构：

[1] Univ Buenos Aires, Fac Ciencias Exactas & Nat, Dept Quim Organ, PROPLAME CONICET, RA-1428 Buenos Aires, DF, Argentina

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2000年 / 43卷 / 01期

关键词：

8-[B-10]- dihydroxyborylharmine; preparation and characterization; boron neutron capture therapy;

D O I：

暂无

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

The preparation and spectral properties (MS, IR and NMR) of 8-[B-10]-dihydroxyborylharmine (III) are described. A general synthetic method was developed for an efficient production of boronated harmine; a potential agent for boron neutron capture therapy (BNCT) in brain.

引用

页码：97 / 101

页数：5

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