Development and mechanistic characterization of USP7 deubiquitinase inhibitors

被引：0

作者：

Wertz, Ingrid ^{[1
]}

Kategaya, Lorna ^{[1
]}

Di Lello, Paola ^{[1
]}

Rouge, Lionel ^{[1
]}

Pastor, Richard ^{[1
]}

Clark, Kevin R. ^{[1
]}

Drummond, Jason ^{[1
]}

Kleinheinz, Tracy ^{[1
]}

Lin, Eva ^{[1
]}

Upton, John-Paul ^{[1
]}

Prakash, Sumit ^{[1
]}

Heideker, Johanna ^{[1
]}

McCleland, Mark ^{[1
]}

Ritorto, Maria Stella ^{[2
]}

Alessi, Dario R. ^{[2
]}

Trost, Matthias ^{[3
]}

Bainbridge, Travis W. ^{[1
]}

Kwok, Michael C. ^{[1
]}

Ma, Taylur P. ^{[1
]}

Stiffler, Zachary ^{[4
]}

Brasher, Bradley ^{[4
]}

Tang, Yinyan ^{[5
]}

Jaishanker, Priya ^{[5
]}

Hearn, Brian ^{[5
]}

Renslo, Adam R. ^{[5
]}

Arkin, Michelle R. ^{[5
]}

Cohen, Frederick ^{[1
]}

Yu, Kebing ^{[1
]}

Peale, Frank ^{[1
]}

Gnad, Florian ^{[1
]}

Chang, Matthew T. ^{[1
]}

Klijn, Christiaan ^{[1
]}

Blackwood, Elizabeth ^{[1
]}

Martin, Scott E. ^{[1
]}

Forrest, William F. ^{[1
]}

Ernst, James A. ^{[1
]}

Ndubaku, Chudi ^{[1
]}

Wang, Xiaojing ^{[1
]}

Beresini, Maureen H. ^{[1
]}

Tsui, Vickie ^{[1
]}

Schwerdtfeger, Carsten ^{[4
]}

Blake, Robert A. ^{[1
]}

Murray, Jeremy ^{[1
]}

Maurer, Till ^{[1
]}

机构：

[1] Genentech Inc, San Francisco, CA 94080 USA

[2] Univ Dundee, Dundee, Scotland

[3] Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, England

[4] Boston Biochem, Cambridge, MA USA

[5] Univ Calif San Francisco, San Francisco, CA 94143 USA

来源：

CANCER RESEARCH | 2018年 / 78卷 / 13期

关键词：

D O I：

10.1158/1538-7445.AM2018-SY23-03

中图分类号：

R73 [肿瘤学];

学科分类号：

100214 ;

摘要：

SY23-03

引用

页数：2

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