Reaction of 2-amino-3-cyano-4,5,6,7-tetrahydrobenzo-[b]thiophene with ethyl acetoacetate:: Novel syntheses of pyridines, pyrazoles, and their fused derivatives

被引：10

作者：

Mohareb, RM ^{[1
]}

Mohamed, MH ^{[1
]}

机构：

[1] Cairo Univ, Fac Sci, Dept Chem, Giza, Egypt

来源：

HETEROATOM CHEMISTRY | 2001年 / 12卷 / 06期

关键词：

D O I：

10.1002/hc.1079

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The reaction of 2-amino-3-cyano-4,5, 6,7-tetrahydrobenzo[b]thiophene 1 with ethyl acetoacetate 2 gave compound 3. The reactivity of the latter product toward a variety of chemical reagents,vas studied to give fused thiophene derivatives of potential pharmaceutical interest. (C) 2001 John Wiley & Sons, Inc.

引用

页码：518 / 527

页数：10

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