Mass Balance and Metabolism of the Taxane Analog [14C]BMS-275183 Following Oral Administration to Humans

被引:0
|
作者
Coemezoglu, S. Nilguen [1 ]
Ly, Van T. [1 ]
Ekhato, Ihoezo V. [2 ]
Gan, Jinping [1 ]
Alland, Leila [3 ]
Humphreys, W. Griff [1 ]
机构
[1] Bristol Myers Squibb Co, PCO Biotransformat, Princeton, NJ USA
[2] Bristol Myers Squibb Co, Chem Synth, Princeton, NJ USA
[3] Bristol Myers Squibb Co, Discovery Med & Clin Pharmacol, Princeton, NJ USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:227 / 228
页数:2
相关论文
共 50 条
  • [1] Metabolism of the taxane analog [14C]BMS-275183 following oral administration to rats and dogs
    Ly, Van T.
    Comezoglu, Nigun
    Zhang, Donglu
    Humphreys, W. Griffith
    Ekhato, Ihoezo V.
    DRUG METABOLISM REVIEWS, 2006, 38 : 178 - 178
  • [2] Metabolism of [14C]BMS-275183 in mouse, rat, dog, monkey and human liver microsomes
    Comezoglu, N
    Kim-Kang, H
    Ogan, M
    Everett, DW
    DRUG METABOLISM REVIEWS, 2002, 34 : 65 - 65
  • [3] Disposition, metabolism and mass balance of [14C]apremilast following oral administration
    Hoffmann, Matthew
    Kumar, Gondi
    Schafer, Peter
    Cedzik, Dorota
    Capone, Lori
    Fong, Kei-Lai
    Gu, Zheming
    Heller, Dennis
    Feng, Hao
    Surapaneni, Sekhar
    Laskin, Oscar
    Wu, Anfan
    XENOBIOTICA, 2011, 41 (12) : 1063 - 1075
  • [4] Disposition, metabolism and mass balance of [14C]apremilast following oral administration
    Hoffmann, M.
    Kumar, G.
    Schafer, P.
    Cedzik, D.
    Capone, L.
    Fong, K.
    Gu, Z.
    Heller, D.
    Feng, H.
    Surapaneni, S.
    Laskin, O.
    Wu, A.
    JOURNAL OF INVESTIGATIVE DERMATOLOGY, 2011, 131 : S89 - S89
  • [5] Biotransformation of [14C]BMS-275183 in bile-duct cannulated (BDC) rats
    Comezoglu, N
    Kim-Kang, H
    Ogan, M
    Everett, DW
    DRUG METABOLISM REVIEWS, 2002, 34 : 65 - 65
  • [6] Absorption, metabolism and excretion of [14C]pomalidomide in humans following oral administration
    Matthew Hoffmann
    Claudia Kasserra
    Josephine Reyes
    Peter Schafer
    Jolanta Kosek
    Lori Capone
    Anastasia Parton
    Heasook Kim-Kang
    Sekhar Surapaneni
    Gondi Kumar
    Cancer Chemotherapy and Pharmacology, 2013, 71 : 489 - 501
  • [7] Absorption, metabolism and excretion of [14C]pomalidomide in humans following oral administration
    Hoffmann, Matthew
    Kasserra, Claudia
    Reyes, Josephine
    Schafer, Peter
    Kosek, Jolanta
    Capone, Lori
    Parton, Anastasia
    Kim-Kang, Heasook
    Surapaneni, Sekhar
    Kumar, Gondi
    CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2013, 71 (02) : 489 - 501
  • [8] A phase I trial investigating a twice weekly administration of the oral taxane BMS-275183 in patients with advanced solid tumors.
    Broker, LE
    Ruyter, R
    Voi, M
    Woo, M
    Astier, L
    Heath, E
    Lorusso, PM
    Giaccone, G
    JOURNAL OF CLINICAL ONCOLOGY, 2005, 23 (16) : 145S - 145S
  • [9] HUMAN MASS BALANCE WITH [14C]-BILASTINE FOLLOWING ORAL ADMINISTRATION TO HEALTHY VOLUNTEERS
    Sologuren, A.
    Lucero, M. L.
    Valiente, R.
    Charles, H.
    Mair, S. J.
    BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2009, 105 : 106 - 107
  • [10] Mass balance study of [14C] rabeprazole following oral administration in healthy subjects
    Setoyama, T.
    Drijfhout, W. J.
    de Merbel, N. C. van
    Humphries, T. J.
    Hasegawa, J.
    INTERNATIONAL JOURNAL OF CLINICAL PHARMACOLOGY AND THERAPEUTICS, 2006, 44 (11) : 557 - 565