An efficient one-pot synthesis of substituted 2-arylbenzo[b]thiophene derivatives

被引：18
|
作者：
Patel, MV [1 ]
Rohde, JJ [1 ]
Gracias, V [1 ]
Kolasa, T [1 ]
机构：
[1] Abbott Labs, Abbott Pk, IL 60064 USA
来源：
TETRAHEDRON LETTERS | 2003年 / 44卷 / 35期
关键词：
D O I：
10.1016/S0040-4039(03)01632-0
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
This communication describes an efficient one-pot procedure for the synthesis of 2-arylbenzo[b]thiophene derivatives via reaction of o-halo or nitro aryl carbonyl compounds with benzyl mercaptans in the presence of an excess of anhydrous K2CO3 at elevated temperature. (C) 2003 Elsevier Ltd. All rights reserved.
引用
收藏
页码：6665 / 6667
页数：3
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