Solid-phase synthesis of head and tail bis-acridinylated peptides

被引:14
|
作者
Sebestík, J
Matejka, P
Hlavácek, J
Stibor, I
机构
[1] Acad Sci Czech Republ, Inst Organ Chem & Biochem, CR-16610 Prague, Czech Republic
[2] Inst Chem Technol, CR-16628 Prague, Czech Republic
关键词
9-amino acridine; solid-phase synthesis; head and tail peptide conjugates;
D O I
10.1016/j.tetlet.2003.11.139
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Amino-acridine conjugates play an important role as biochemical probes and/or drugs. Solid-phase synthesis of such compounds suitable for library construction and biological screening is described. (C) 2003 Elsevier Ltd. All rights reserved.
引用
收藏
页码:1203 / 1205
页数:3
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